SCHEMBL5405545

SCHEMBL5405545

CCOc1cc(C#N)ccc1CBr

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.54
HTR2A P28223 1/20 0.39
KCNH2 Q12809 1/20 0.39
GRM5 P41594 1/20 0.39
S1PR1 P21453 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
AGPAT2 O15120 2/20 0.38
GABRG2 P18507 1/20 0.37
GABRB3 P28472 1/20 0.37
GABRA5 P31644 1/20 0.37
GABRA3 P34903 1/20 0.37
DRD4 P21917 1/20 0.37
PDE5A O76074 1/20 0.36
CYP2A6 P11509 1/20 0.36
GAA P10253 1/20 0.36
AR P10275 3/20 0.36
NR3C2 P08235 2/20 0.35
NR3C1 P04150 1/20 0.35
PGR P06401 1/20 0.35
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6476469 0.83 TRPV4 (0.54) TRPV4HTR2AKCNH2GRM5S1PR1
SCHEMBL14468631 0.83 TRPV4 (0.54) TRPV4HTR2AKCNH2GRM5S1PR1
SCHEMBL411153 0.83 AR (0.47) TRPV4HTR2AKCNH2GAAAR
Hydrochloric Acid SCHEMBL6476582 0.82 TRPV4 (0.52) TRPV4HTR2AKCNH2GRM5S1PR1
SCHEMBL8735777 0.81 TRPV4 (0.51) TRPV4HTR2AKCNH2GRM5S1PR1
SCHEMBL27001729 0.81 CYP19A1 (0.41) TRPV4HTR2AKCNH2ARALDH1A1
SCHEMBL1664918 0.81 TRPV4 (0.51) TRPV4HTR2AKCNH2GRM5S1PR1
SCHEMBL1402437 0.80 TRPV4 (0.61) TRPV4GRM5S1PR1GABRG2GABRB3
SCHEMBL5900831 0.80 KCNH2 (0.42) TRPV4HTR2AKCNH2S1PR1AR
SCHEMBL14468537 0.80 TRPV4 (0.54) TRPV4HTR2AKCNH2GRM5S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7241625-B2 Carbonyl compound scavenger and method of quantifying carbonyl compound using the same SUMIKA CHEMICAL ANALYSIS SERVICE, LIMITED (JP) 2007-07-10 US disclosed
US-7241625-B2 Carbonyl compound scavenger and method of quantifying carbonyl compound using the same SUMIKA CHEMICAL ANALYSIS SERVICE, LIMITED (JP) 2007-07-10 US disclosed
US-20060275913-A1 Carbonyl compound scavenger and method of quantifying carbonyl compound using the same SUMIKA CHEMICAL ANALYSIS SERVICE, LIMITED (JP) 2006-12-07 US disclosed
US-6900319-B2 Thrombin inhibitors ABBOTT GMBH & CO. KG (DE) 2005-05-31 US disclosed
US-20020169318-A1 Novel thrombin inhibitors ABBVIE DEUTSCHLAND GMBH & CO KG (DE) 2002-11-14 US disclosed
US-6444817-B1 ANTICOAGULANTS ABBOTT LABORATORIES 2002-09-03 US disclosed
US-6030972-A 2- OR 5-AMINOMETHYL,2- OR 5-CYANOPYRIMIDINES AS INTERMEDIATES OF ANTICOAGULANTS IN EXTRACORPOREAL CIRCULATION (HEART-LUNG MACHINE, HEMODIALYSIS) BASF AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed
EP-0873356-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1998-10-28 EP disclosed
WO-1996025426-A1 NOVEL DIPEPTIDE AMIDINES AS THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 1996-08-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060275913-A1 Carbonyl compound scavenger and method of quantifying carbonyl compound using the same CBR1, CBR3, HAO2 TRPV4 531/4885HTR2A 3433/4885KCNH2 99/4885
US-20020169318-A1 Novel thrombin inhibitors TFPI, SERPINC1, F11 TRPV4 4468/4885HTR2A 3737/4885KCNH2 3150/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.