SCHEMBL5406058

SCHEMBL5406058

COc1cncc(C(C)=CCCN)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 2/20 0.38
MKNK1 Q9BUB5 1/20 0.38
CYP11B1 P15538 4/20 0.36
CYP11B2 P19099 4/20 0.36
MAP4K4 O95819 2/20 0.36
ROCK2 O75116 1/20 0.36
PRKACA P17612 1/20 0.36
ROCK1 Q13464 1/20 0.36
DYRK1A Q13627 1/20 0.36
NTRK3 Q16288 1/20 0.36
PKN2 Q16513 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
STK17A Q9UEE5 1/20 0.36
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
TBXAS1 P24557 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7744105 0.85 CYP11B1 (0.40) MKNK2CYP11B1CYP11B2MAP4K4ROCK2
SCHEMBL8590780 0.80 KDM4E (0.44) TBXAS1
SCHEMBL365734 0.79 MKNK2 (0.37) MKNK2MKNK1CYP11B1CYP11B2MAP4K4
SCHEMBL7071083 0.78 MKNK2 (0.35) MKNK2MKNK1CYP11B1CYP11B2MAP4K4
SCHEMBL7738084 0.75 TBXAS1 (0.38) TBXAS1
SCHEMBL5196886 0.74 AOC3 (0.34) TBXAS1
SCHEMBL7238664 0.71 MKNK1 (0.49) MKNK2MKNK1CYP11B1CYP11B2MAP4K4
SCHEMBL3956347 0.71 MKNK1 (0.33) MKNK2MKNK1
Hydrochloric Acid SCHEMBL7240593 0.70 MKNK1 (0.48) MKNK2MKNK1CYP11B1CYP11B2MAP4K4
SCHEMBL3128200 0.70 TBXAS1 (0.61) CYP1A2CYP3A4TBXAS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-3899126-B2 2007-03-28 JP claimed
JP-2001520628-A 2001-10-30 JP claimed
EP-0801527-A4 PHARMACEUTICAL COMPOSITIONS FOR PREVENTION AND TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS REYNOLDS TOBACCO CO R (US) 2001-09-05 EP claimed
EP-0801527-A1 PHARMACEUTICAL COMPOSITIONS FOR PREVENTION AND TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS R.J. REYNOLDS TOBACCO COMPANY (US) 1997-10-22 EP claimed
WO-1996020600-A1 PHARMACEUTICAL COMPOSITIONS FOR PREVENTION AND TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS R.J. REYNOLDS TOBACCO COMPANY (US) 1996-07-11 WO claimed