SCHEMBL5450814

SCHEMBL5450814

C[C@@]12CCC[C@H]1[C@@H]1CCC3CC=CC[C@]3(C)[C@H]1CC2

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 5/20 0.59
NR1I3 Q14994 2/20 0.55
CDK5 Q00535 1/20 0.55
CDK5R1 Q15078 1/20 0.55
GRIN1 Q05586 7/20 0.47
GRIN2B Q13224 7/20 0.47
MBOAT4 Q96T53 3/20 0.45
ALDH1A1 P00352 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2955007 1.00 CYP19A1 (0.59) CYP19A1NR1I3CDK5CDK5R1GRIN1
SCHEMBL10609022 0.81 CDK5 (0.44) CYP19A1NR1I3CDK5CDK5R1GRIN1
SCHEMBL3224692 0.80 CDK5 (0.43) CYP19A1NR1I3CDK5CDK5R1GRIN1
SCHEMBL10609234 0.80 CDK5 (0.43) CYP19A1NR1I3CDK5CDK5R1GRIN1
SCHEMBL10780071 0.80 CDK5 (0.43) CYP19A1NR1I3CDK5CDK5R1GRIN1
SCHEMBL11654859 0.80 NR1I3 (0.46) CYP19A1NR1I3CDK5CDK5R1GRIN1
SCHEMBL1319449 0.79 NR1I3 (0.58) CYP19A1NR1I3CDK5CDK5R1GRIN1
SCHEMBL1319450 0.79 NR1I3 (0.58) CYP19A1NR1I3CDK5CDK5R1GRIN1
SCHEMBL19733225 0.79 NR1I3 (0.58) CYP19A1NR1I3CDK5CDK5R1GRIN1
SCHEMBL10879635 0.79 CYP19A1 (0.55) CYP19A1NR1I3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20220193095-A9 PHARMACEUTICAL COMPOSITIONS Shenzhen Pharmacin Co., Ltd. (CN) 2022-06-23 US claimed
US-20220193095-A9 PHARMACEUTICAL COMPOSITIONS Shenzhen Pharmacin Co., Ltd. (CN) 2022-06-23 US disclosed
US-20220133749-A1 METHODS AND COMPOSITIONS FOR TREATING CANCER JANSSEN ONCOLOGY INC (US) 2022-05-05 US disclosed
US-20070111973-A1 TREATMENT OF TUMOURS HAGSTROM TOMAS 2007-05-17 US disclosed
US-20050192262-A1 Treatment of tumours HAGSTROM, TOMAS (SE) 2005-09-01 US disclosed
EP-1379542-A2 TREATMENT OF TUMOURS Hagström, Tomas (SE) 2004-01-14 EP disclosed
WO-2002072003-A2 USE OF STEROID DERIVATIVES FOR THE TREATMENT OF A BENIGHN AND/OR MALIGNANT TUMOUR HAGSTROEM TOMAS (SE) 2002-09-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050192262-A1 Treatment of tumours SULT2A1, SULT1A1, HSD17B11 CYP19A1 20/4885NR1I3 134/4885CDK5 238/4885
US-20220193095-A9 PHARMACEUTICAL COMPOSITIONS LIPA, LIPC, MGLL CYP19A1 674/4885NR1I3 3198/4885CDK5 4709/4885
US-20220133749-A1 METHODS AND COMPOSITIONS FOR TREATING CANCER CYP17A1, HSD17B7, HSD17B11 CYP19A1 17/4885NR1I3 600/4885CDK5 291/4885
US-20070111973-A1 TREATMENT OF TUMOURS SULT2A1, SULT1A1, SULT1E1 CYP19A1 24/4885NR1I3 139/4885CDK5 312/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.