SCHEMBL5458774

SCHEMBL5458774

CS(=O)(=O)c1ccc(Nc2ccc(C#N)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.57
CA1 P00915 3/20 0.50
CA2 P00918 3/20 0.50
KDM1A O60341 1/20 0.49
IDO1 P14902 3/20 0.49
CA12 O43570 2/20 0.49
CA9 Q16790 2/20 0.49
PIP4K2A P48426 1/20 0.47
SIRT2 Q8IXJ6 1/20 0.46
CYP19A1 P11511 2/20 0.45
DHODH Q02127 1/20 0.44
IKBKB O14920 1/20 0.44
CYP11B1 P15538 1/20 0.44
CYP11B2 P19099 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL803901 0.88 PTGS2 (0.68) PTGS2CA1CA2KDM1ACA12
SCHEMBL25667539 0.84 ENPP2 (0.54) CA1CA2CA12CA9PIP4K2A
SCHEMBL4190362 0.82 PTGS2 (0.72) PTGS2CA1CA2CA12CA9
SCHEMBL4187483 0.82 ALPL (0.49) PTGS2CA1CA2CA12CA9
SCHEMBL27888182 0.81 CA1 (0.71) CA1CA2CA12CA9IKBKB
SCHEMBL27374894 0.81 SOS1 (0.51) PTGS2PIP4K2A
SCHEMBL30751412 0.81 SOS1 (0.51) PTGS2PIP4K2A
SCHEMBL395539 0.79 CA2 (0.52) CA1CA2IDO1CA12CA9
SCHEMBL10951291 0.78 PTGS2 (0.57) PTGS2CA1CA2CA12CA9
SCHEMBL17492799 0.77 MAPT (0.49) CA1CA2CA12SIRT2CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070129433-A1 Diphenylamine derivatives MERCK PATENT GMBH (DE) 2007-06-07 US claimed
EP-1687253-A2 DIPHENYLAMINE DERIVATIVES Merk Patent Gmbh (DE) 2006-08-09 EP claimed
WO-2005051888-A2 DIPHENYLAMINE DERIVATIVES MERK PATENT GMBH (DE) 2005-06-09 WO claimed
US-20070129433-A1 Diphenylamine derivatives MERCK PATENT GMBH (DE) 2007-06-07 US disclosed
US-20070129433-A1 Diphenylamine derivatives MERCK PATENT GMBH (DE) 2007-06-07 US disclosed
US-20070123586-A1 Nitroso derivatives of diphenylamine MERCK PATENT GMBH (DE) 2007-05-31 US disclosed
US-20070123586-A1 Nitroso derivatives of diphenylamine MERCK PATENT GMBH (DE) 2007-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070123586-A1 Nitroso derivatives of diphenylamine NOS3, CBR3, CBR1 PTGS2 580/4885CA1 2615/4885CA2 1737/4885
US-20070129433-A1 Diphenylamine derivatives CCNY, CHKB, CHKA PTGS2 4190/4885CA1 1145/4885CA2 346/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.