SCHEMBL5484256

SCHEMBL5484256

NCC(O)CN(C(CS(=O)(=O)Cc1ccccc1C(N)=O)C(=O)NCC(=O)CNS(=O)(=O)c1ccccc1)S(=O)(=O)c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.33
CTSS P25774 1/20 0.33
KCNA5 P22460 1/20 0.32
KAT6A Q92794 1/20 0.31
MMP2 P08253 1/20 0.30
MMP9 P14780 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5440671 0.71 MMP1 (0.36) KCNA5KAT6AMMP2MMP9
SCHEMBL5484261 0.67 CA2 (0.34) CTSKCTSSMMP2MMP9
SCHEMBL5440673 0.66 LARS1 (0.41) CTSKCTSSMMP2MMP9
SCHEMBL6557593 0.63 KEAP1 (0.41) CTSKCTSSMMP2MMP9
SCHEMBL5440888 0.59 GBA1 (0.63) MMP2MMP9
SCHEMBL5471723 0.59 PRMT1 (0.40) CTSKCTSSMMP2MMP9
SCHEMBL740682 0.58 KMT2A (0.51)
SCHEMBL28880375 0.58 KDM4E (0.42)
SCHEMBL2969958 0.57 MMP1 (0.59) MMP2MMP9
SCHEMBL6401361 0.55 MAPT (0.52)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7196099-B2 Compounds and compositions as cathepsin inhibitors AVENTIS PHARMACEUTICALS INC. (US) 2007-03-27 US disclosed