SCHEMBL5484261

SCHEMBL5484261

NC(CS(=O)(=O)Cc1ccccc1)C(=O)NCC(=O)CNS(=O)(=O)c1ccccc1.NCC(O)Cc1ccccc1S(N)(=O)=O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 5/20 0.34
CTSK P43235 2/20 0.32
CTSS P25774 1/20 0.32
CA1 P00915 3/20 0.32
CA12 O43570 2/20 0.32
LIPC P11150 1/20 0.31
LIPG Q9Y5X9 1/20 0.31
HPGD P15428 1/20 0.31
LARS1 Q9P2J5 1/20 0.31
GBA1 P04062 1/20 0.31
CA9 Q16790 1/20 0.31
HSD17B10 Q99714 1/20 0.30
CASP1 P29466 1/20 0.30
PTGES2 Q9H7Z7 1/20 0.30
ALDH1A1 P00352 1/20 0.30
MMP1 P03956 1/20 0.30
MMP2 P08253 1/20 0.30
MMP3 P08254 1/20 0.30
MMP7 P09237 1/20 0.30
MMP9 P14780 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5440673 0.85 LARS1 (0.41) CTSKCTSSLARS1GBA1CASP1
SCHEMBL6557593 0.68 KEAP1 (0.41) CTSKCTSSGBA1CASP1ALDH1A1
SCHEMBL5484256 0.67 CTSK (0.33) CTSKCTSSMMP2MMP9
SCHEMBL5441961 0.65 CA2 (0.41) CA2CA1CA12CA9ALDH1A1
SCHEMBL6843005 0.64 CTSS (0.53) CTSKCTSSHSD17B10ALDH1A1
SCHEMBL14491115 0.64 CTSS (0.53) CTSKCTSSHSD17B10ALDH1A1
SCHEMBL6742782 0.64 CTSC (0.49) CTSKCTSSHPGD
SCHEMBL5471723 0.64 PRMT1 (0.40) CTSKCTSSCASP1ALDH1A1MMP1
SCHEMBL6742169 0.62 CTSC (0.47) CTSKCTSSHPGD
SCHEMBL6742769 0.62 CTSC (0.47) CTSKCTSSHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7196099-B2 Compounds and compositions as cathepsin inhibitors AVENTIS PHARMACEUTICALS INC. (US) 2007-03-27 US disclosed