SCHEMBL5486403

SCHEMBL5486403

CN(C(=O)c1cccnc1)c1ccc(NC2CCOCC2)nc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.46
HSD17B10 Q99714 5/20 0.43
MAPK1 P28482 2/20 0.43
TP53 P04637 2/20 0.43
USP2 O75604 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
KCNH2 Q12809 6/20 0.41
ATM Q13315 3/20 0.41
ATR Q13535 1/20 0.41
PLOD2 O00469 1/20 0.40
PLOD3 O60568 1/20 0.40
PLOD1 Q02809 1/20 0.40
KDM4E B2RXH2 3/20 0.39
ALDH1A1 P00352 1/20 0.39
FYN P06241 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5486419 0.79 CYP2C19 (0.58) TP53ALOX15KDM4EALDH1A1NPC1
SCHEMBL5083468 0.70 ALDH1A1 (0.65) TP53TSHRALDH1A1RAB9ASMN1; SMN2
SCHEMBL28630199 0.70 MLYCD (0.65) MLYCDHSD17B10MAPK1TP53USP2
SCHEMBL5935115 0.69 MLYCD (0.67) MLYCDHSD17B10MAPK1TP53USP2
SCHEMBL4735448 0.68 MAPK14 (0.55) TP53TSHRALDH1A1HCAR3SMN1; SMN2
SCHEMBL22983342 0.68 ALDH1A1 (0.65) MLYCDHSD17B10TP53NPSR1KDM4E
Water SCHEMBL11233247 0.68 MLYCD (0.62) MLYCDHSD17B10MAPK1TP53USP2
Water SCHEMBL11233238 0.68 MLYCD (0.62) MLYCDHSD17B10MAPK1TP53USP2
SCHEMBL789922 0.67 ALDH1A1 (0.53) HSD17B10TP53ALOX15KDM4EALDH1A1
SCHEMBL5486398 0.67 CYP1A2 (0.46) MAPK1TP53TSHRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007056016-A2 BISAMIDE CYTOKINE INHIBITORS KEMIA, INC. (US) 2007-05-18 WO disclosed