SCHEMBL5486423

SCHEMBL5486423

Cc1cc2c(cc1-c1cc(CN3C(=O)CSC3=O)ccc1OC(F)(F)F)C(C)(C)CCC2(C)C

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
RXRA P19793 17/20 0.49
KCNN4 O15554 2/20 0.42
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7459610 0.93 KCNN4 (0.43) RXRAKCNN4POLB
SCHEMBL7464760 0.84 KCNN4 (0.42) KCNN4POLB
SCHEMBL7460353 0.84 GSK3A (0.48) RXRAKCNN4POLB
SCHEMBL7466491 0.84 POLB (0.43) RXRAKCNN4POLB
SCHEMBL7468575 0.83 KMT2A (0.46) RXRAPOLB
SCHEMBL7459835 0.83 KCNN4 (0.42) KCNN4POLB
SCHEMBL5485145 0.82 RXRA (0.46) RXRAPOLB
SCHEMBL5491294 0.82 KCNN4 (0.43) RXRAKCNN4POLB
SCHEMBL7461597 0.82 KCNN4 (0.41) RXRAKCNN4
SCHEMBL7463442 0.81 ALDH1A1 (0.46) RXRAKCNN4POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7226940-B2 Substituted heterocycles for the treatment of diabetes and other diseases INCYTE SAN DIEGO, INC. (US) 2007-06-05 US disclosed
US-20060004059-A1 Substituted heterocycles for the treatment of diabetes and other diseases PFAHL MAGNUS 2006-01-05 US disclosed
US-6515003-B1 Useful in the treatment of diseases related to lipid and carbohydrate metabolism MAXIA PHARMACEUTICALS, INC. 2003-02-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060004059-A1 Substituted heterocycles for the treatment of diabetes and other diseases FABP4, HPGDS, GPR119 RXRA 307/4885KCNN4 4620/4885POLB 3245/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.