SCHEMBL549252

SCHEMBL549252

Fc1ccc2c(c1)NCC2

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 6/20 0.56
PARP1 P09874 5/20 0.56
HTR2C P28335 3/20 0.44
HTR2A P28223 1/20 0.44
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
GFER P55789 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HTR5A P47898 2/20 0.42
P4HB P07237 1/20 0.40
PYGL P06737 1/20 0.39
GRM5 P41594 2/20 0.39
PARP11 Q9NR21 1/20 0.39
HTR2B P41595 2/20 0.39
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
F7 P08709 1/20 0.35
F3 P13726 1/20 0.35
DPP4 P27487 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30583047 1.00 PARP10 (0.56) PARP10PARP1HTR2CHTR2ADRD2
SCHEMBL29622425 0.88 PYGL (0.49) PARP10PARP1HTR2CHTR2AGFER
SCHEMBL3112268 0.88 PYGL (0.49) PARP10PARP1HTR2CHTR2AGFER
Hydrochloric Acid SCHEMBL30142485 0.86 PYGL (0.48) PARP10PARP1HTR2CHTR2AGFER
Hydrochloric Acid SCHEMBL2144161 0.86 PYGL (0.48) PARP10PARP1HTR2CHTR2AGFER
SCHEMBL5467312 0.86 PYGL (0.45) PARP10PARP1HTR2CHTR2AGFER
SCHEMBL549063 0.83 DRD2 (0.59) PARP10PARP1HTR2CHTR2ADRD2
SCHEMBL23188859 0.81 PARP10 (0.56) PARP10PARP1HTR2CHTR2ASMN1; SMN2
SCHEMBL9081400 0.81 PARP1 (0.44) PARP10PARP1HTR2CHTR2ADRD2
Hydrochloric Acid SCHEMBL17799458 0.81 DRD2 (0.57) PARP10PARP1HTR2CHTR2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 245 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115353478-A Preparation method of indole compound 南京工业大学 2022-11-18 CN claimed
WO-2026103853-A1 TSHR ANTAGONIST COMPOUND, PHARMACEUTICAL COMPOSITION, METHOD FOR PREPARING SAME, AND USE THEREOF 长春金赛药业有限责任公司 2026-05-21 WO disclosed
US-12612424-B2 HPK1 inhibitors and uses thereof REGOR PHARMACEUTICALS, INC. (US) 2026-04-28 US disclosed
EP-4605089-A1 COMPOUNDS USEFUL IN MODULATING EGFR AND PI3K Mekanistic Therapeutics LLC (US) 2025-08-27 EP disclosed
US-20250171420-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME MONTE ROSA THERAPEUTICS AG (CH) 2025-05-29 US disclosed
EP-4301739-B1 FPR2 (FORMYL PEPTIDE RECEPTOR 2) RECEPTOR AGONISTS AND THEIR USE IN THE TREATMENT OF THE AUTISM SPECTRUM DISORDER UNIV DEGLI STUDI DI BARI ALDO MORO (IT) 2025-04-23 EP disclosed
EP-4540240-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME Monte Rosa Therapeutics AG (CH) 2025-04-23 EP disclosed
EP-4536363-A1 SULFAMIDE DERIVATIVES AS CYCLIN-DEPENDENT KINASE 2 INHIBITORS Nikang Therapeutics, Inc. (US) 2025-04-16 EP disclosed
CN-119822910-A Method for catalyzing heterogeneous reduction of nitrogen-containing heterocyclic compound by using magnesium metal 延安大学 2025-04-15 CN disclosed
CN-113227054-B ROCK kinase inhibitors 切尔韦洛治疗有限责任公司 2025-04-11 CN disclosed
EP-1266896-A1 Linear ou cyclic ureas, process for their preparation and pharmaceutical compositions containing them Les Laboratoires Servier (FR) 2002-12-18 EP disclosed
US-20010009911-A1 New linear or cyclic ureas LES LABORATOIRES SERVIER (FR) 2001-07-26 US disclosed
EP-1113014-A1 Linear or cyclic ureas, a process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 2001-07-04 EP disclosed
US-5981752-A Tricyclic compounds having fungicidal activity, their preparation and their use SANKYO COMPANY, LIMITED (JP) 1999-11-09 US disclosed
US-5773618-A PYRROLOQUINOLINONE DERIVATIVES SANKYO COMPANY, LIMITED (JP) 1998-06-30 US disclosed
US-5736534-A HYPERPROLIFERATIVE DISEASES; INHIBITORS OF PROTEIN-TYROSINE KINASES SUCH AS EPIDERMAL GROWTH FACTOR RECEPTOR; BRAIN, LUNG, BREAST CANCER; PSORIASIS AND BENIGN PROSTATE HYPERPLASIA PFIZER INC. (US) 1998-04-07 US disclosed
EP-0807631-A1 Tricyclic compounds having fungicidal activity, their preparation and their use SANKYO COMPANY LIMITED (JP) 1997-11-19 EP disclosed
EP-0746554-A1 4-HETEROCYCLYL-SUBSTITUTED QUINAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS ANTI-CANCER AGENTS PFIZER INC. (US) 1996-12-11 EP disclosed
WO-1995023141-A1 4-HETEROCYCLYL-SUBSTITUTED QUINAZOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS ANTI-CANCER AGENTS PFIZER INC. (US) 1995-08-31 WO disclosed
US-4904684-A 2-(4,5-dihydro-1H-imidazol-2-yl)-1,2,4,5-tetrahydropyrrolo[3,2,1-hi]indole derivatives useful as antidiabetic agents SYNTHELABO (FR) 1990-02-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20010009911-A1 New linear or cyclic ureas GUCY1B1, UACA, LIPG PARP10 4220/4885PARP1 3068/4885HTR2C 1972/4885
US-12612424-B2 HPK1 inhibitors and uses thereof NEK11, NEK1, CSNK1A1 PARP10 810/4885PARP1 1017/4885HTR2C 2173/4885
US-20250171420-A1 MOLECULAR GLUE DEGRADERS AND METHODS OF USING THE SAME PSMA1, CSNK1G1, CSNK1A1 PARP10 705/4885PARP1 307/4885HTR2C 4347/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.