SCHEMBL5499274

SCHEMBL5499274

CCCc1c([N+](=O)[O-])cc2c(c1F)NC(=O)C2

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 4/20 0.35
PGR P06401 2/20 0.33
MAPT P10636 2/20 0.33
ALDH1A1 P00352 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
GAA P10253 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5502610 0.90 TDP2 (0.36) TDP2PGRMAPTALDH1A1TDP1
SCHEMBL5498328 0.88 TDP2 (0.35) TDP2PGRCYP11B1CYP11B2
SCHEMBL5504412 0.81 TDP2 (0.34) TDP2PGRCYP11B1CYP11B2
SCHEMBL5499002 0.80 TDP2 (0.38) TDP2PGRALDH1A1TDP1CYP11B1
SCHEMBL5502598 0.79 AHR (0.30) TDP2
SCHEMBL5504827 0.76 TDP2 (0.36) TDP2PGRTDP1CYP11B1CYP11B2
SCHEMBL5503483 0.74 TDP2 (0.36) TDP2PGRCYP11B1CYP11B2
SCHEMBL5498169 0.72 PGR (0.41) TDP2PGRALDH1A1TDP1GAA
SCHEMBL3139883 0.72 TDP2 (0.41) TDP2PGRMAPTALDH1A1TDP1
SCHEMBL5501936 0.70 AHR (0.32) TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869030-A1 7-FLUORO-1,3-DIHYDRO-INDOL-2-ONE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS Pharmacia & Upjohn Company LLC (US) 2007-12-26 EP disclosed
EP-1781642-A1 OXAZOLIDINONES CONTAINING OXINDOLES AS ANTIBACTERIAL AGENTS Pharmacia & Upjohn Company LLC (US) 2007-05-09 EP disclosed
EP-1781643-A1 OXINDOLE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS Pharmacia & Upjohn Company LLC (US) 2007-05-09 EP disclosed
WO-2006106427-A1 7-FLUORO-1,3-DIHYDRO-INDOL-2-ONE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-10-12 WO disclosed
WO-2006016220-A1 OXINDOLE OXAZOLIDINONES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-02-16 WO disclosed
WO-2006016221-A1 OXAZOLIDINONES CONTAINING OXINDOLES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-02-16 WO disclosed