SCHEMBL5500299

SCHEMBL5500299

OC1(CCCc2cccc(Cl)c2Cl)CCNCC1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.42
SLC6A2 P23975 5/20 0.39
SLC6A4 P31645 5/20 0.39
PNMT P11086 1/20 0.39
KCNH2 Q12809 2/20 0.36
REN P00797 1/20 0.36
DRD2 P14416 4/20 0.36
DRD3 P35462 3/20 0.36
ADRB1 P08588 1/20 0.36
IDO1 P14902 2/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
SLC6A3 Q01959 4/20 0.34
CYP2D6 P10635 2/20 0.34
ACAT2 Q9BWD1 1/20 0.34
CYP3A4 P08684 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5502511 0.91 TAAR1 (0.45) TAAR1SLC6A2SLC6A4PNMTKCNH2
SCHEMBL5499318 0.86 KCNH2 (0.33) TAAR1SLC6A2SLC6A4KCNH2REN
SCHEMBL5493818 0.86 FFAR4 (0.41) SLC6A2SLC6A4KCNH2RENDRD2
SCHEMBL5500092 0.83 FFAR4 (0.43) SLC6A2SLC6A4KCNH2RENCYP3A4
SCHEMBL5495138 0.80 KCNH2 (0.37) SLC6A2SLC6A4KCNH2RENALDH1A1
SCHEMBL5495293 0.80 P2RX7 (0.38) SLC6A2SLC6A4KCNH2SLC6A3CYP2D6
SCHEMBL5501439 0.77 FFAR4 (0.40) SLC6A2SLC6A4KCNH2RENDRD2
SCHEMBL5498352 0.77 DRD2 (0.34) TAAR1SLC6A2SLC6A4KCNH2REN
SCHEMBL4390004 0.77 FFAR4 (0.39) SLC6A2SLC6A4KCNH2RENDRD2
SCHEMBL5499300 0.74 SLC6A2 (0.45) SLC6A2SLC6A4KCNH2RENCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765779-A1 NEW SUBSTITUTED PIPERIDINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2007-03-28 EP claimed
WO-2005121092-A1 NEW SUBSTITUTED PIPERIDINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2005-12-22 WO claimed
EP-1765779-A1 NEW SUBSTITUTED PIPERIDINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2007-03-28 EP disclosed
WO-2005121092-A1 NEW SUBSTITUTED PIPERIDINES AS MODULATORS OF DOPAMINE NEUROTRANSMISSION A. CARLSSON RESEARCH AB (SE) 2005-12-22 WO disclosed