SCHEMBL5506636

SCHEMBL5506636

COc1ccc2nccc(NC(=O)CCC3CCCN(Cc4ccc5c(c4)OCCO5)C3)c2n1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.56
KDM4E B2RXH2 2/20 0.53
TARDBP Q13148 1/20 0.46
MCHR1 Q99705 6/20 0.42
KMT2A Q03164 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5514123 0.93 KCNH2 (0.55) KCNH2KDM4ETARDBP
SCHEMBL5512371 0.87 KCNH2 (0.58) KCNH2KDM4EMCHR1KMT2A
SCHEMBL5508574 0.77 ALDH1A1 (0.47) MCHR1KMT2A
SCHEMBL5508579 0.77 ALDH1A1 (0.47) MCHR1KMT2A
SCHEMBL14573144 0.76 KCNH2 (0.61) KCNH2
SCHEMBL5509547 0.76 CYP2C9 (0.45) KCNH2KDM4EKMT2A
SCHEMBL5512152 0.75 KDM4E (0.54) KDM4ETARDBPMCHR1KMT2A
SCHEMBL5507933 0.75 KCNH2 (0.45) KCNH2KMT2A
SCHEMBL5764517 0.75 KCNH2 (0.58) KCNH2
SCHEMBL14372272 0.74 KCNH2 (0.62) KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799676-A2 NEW BICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2007-06-27 EP disclosed
WO-2006032466-A2 NEW BICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-30 WO disclosed