SCHEMBL5509547

SCHEMBL5509547

COc1ccc2nccc(NC(=O)CCC3CCCN(C(=O)OC(C)(C)C)C3)c2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.45
CHEK2 O96017 1/20 0.42
GLS O94925 2/20 0.41
KCNH2 Q12809 3/20 0.40
SCN9A Q15858 1/20 0.40
ACKR3 P25106 1/20 0.40
FPR3 P25089 1/20 0.39
FPR2 P25090 1/20 0.39
PIK3CD O00329 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
TP53 P04637 1/20 0.38
TSHR P16473 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
BACE1 P56817 2/20 0.38
CTSD P07339 1/20 0.38
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL634125 0.79 KCNH2 (0.44) KCNH2PIK3CD
SCHEMBL634126 0.79 KCNH2 (0.44) KCNH2PIK3CD
SCHEMBL633007 0.78 KCNH2 (0.50) KCNH2PIK3CDALDH1A1
SCHEMBL5775818 0.78 MAP4K4 (0.45) KCNH2PIK3CDMEN1KMT2AKDM4E
SCHEMBL5511934 0.78 ROCK2 (0.46) KCNH2MEN1KMT2ANPC1TP53
SCHEMBL5508574 0.78 ALDH1A1 (0.47) MEN1KMT2ATSHRALDH1A1
SCHEMBL5508579 0.78 ALDH1A1 (0.47) MEN1KMT2ATSHRALDH1A1
SCHEMBL5507933 0.75 KCNH2 (0.45) KCNH2MEN1KMT2AALDH1A1
SCHEMBL5514123 0.75 KCNH2 (0.55) KCNH2KDM4E
SCHEMBL6221359 0.74 KCNH2 (0.38) KCNH2PIK3CDKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799676-A2 NEW BICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2007-06-27 EP disclosed
WO-2006032466-A2 NEW BICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-30 WO disclosed