SCHEMBL5508574

SCHEMBL5508574

COc1ccc2nccc(NC(=O)CCC3CCCN(C/C=C/c4ccccc4)C3)c2n1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
LMNA P02545 4/20 0.47
MEN1 O00255 6/20 0.46
KMT2A Q03164 6/20 0.46
POLB P06746 1/20 0.41
GAA P10253 2/20 0.41
TSHR P16473 2/20 0.41
MAPK1 P28482 1/20 0.41
MCHR1 Q99705 1/20 0.39
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
USP2 O75604 1/20 0.38
MAPT P10636 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5508579 1.00 ALDH1A1 (0.47) ALDH1A1LMNAMEN1KMT2APOLB
SCHEMBL5507933 0.78 KCNH2 (0.45) ALDH1A1MEN1KMT2ACNR1CNR2
SCHEMBL5509547 0.78 CYP2C9 (0.45) ALDH1A1MEN1KMT2ATSHR
SCHEMBL5506636 0.77 KCNH2 (0.56) KMT2AMCHR1
SCHEMBL5514123 0.76 KCNH2 (0.55)
SCHEMBL5511934 0.75 ROCK2 (0.46) ALDH1A1MEN1KMT2ATSHRCNR1
SCHEMBL14372276 0.73 KCNH2 (0.44) ALDH1A1POLBCNR1CNR2
SCHEMBL5267677 0.72 SLC2A1 (0.47) CNR1CNR2
SCHEMBL5267681 0.72 SLC2A1 (0.47) CNR1CNR2
SCHEMBL5514132 0.72 KCNH2 (0.35) ALDH1A1MEN1KMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799676-A2 NEW BICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2007-06-27 EP claimed
WO-2006032466-A2 NEW BICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-30 WO claimed