SCHEMBL5506908

SCHEMBL5506908

COc1cc(F)c2nccc(C(O)C(O)c3ccccc3)c2c1

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC10A1 Q14973 1/20 0.38
ADAMTS5 Q9UNA0 2/20 0.36
PDE10A Q9Y233 4/20 0.36
RPS6KB1 P23443 4/20 0.36
AURKA O14965 3/20 0.36
CYP3A4 P08684 1/20 0.35
BCHE P06276 1/20 0.34
MCL1 Q07820 1/20 0.34
PDE2A O00408 1/20 0.34
ACHE P22303 1/20 0.33
LMNA P02545 1/20 0.33
CRHR1 P34998 1/20 0.33
ACVR1 Q04771 1/20 0.33
P4HB P07237 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3929993 0.79 ROCK2 (0.35) PDE10ACYP3A4CRHR1ACVR1
SCHEMBL3403559 0.78 NSD2 (0.35) LMNA
SCHEMBL3373217 0.76 CRHR1 (0.36) CYP3A4BCHECRHR1ACVR1
SCHEMBL3452969 0.76 CRHR1 (0.36) CYP3A4BCHECRHR1ACVR1
SCHEMBL2923376 0.74 NOS3 (0.40) PDE10ACYP3A4PDE2ALMNAACVR1
SCHEMBL7140533 0.73 KDM4E (0.35) PDE10APDE2ALMNAACVR1
SCHEMBL4279169 0.71 NOS3 (0.43) PDE10ACYP3A4PDE2AACVR1
SCHEMBL18544288 0.71 CCR1 (0.38) PDE10ACYP3A4PDE2ALMNAACVR1
SCHEMBL3375901 0.71 CCR1 (0.38) PDE10ACYP3A4PDE2ALMNAACVR1
SCHEMBL5505859 0.71 ALK (0.49) CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799676-A2 NEW BICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2007-06-27 EP disclosed
WO-2006032466-A2 NEW BICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-30 WO disclosed