SCHEMBL5507540

SCHEMBL5507540

O=C(c1cccc(F)c1OCC1CC1)C1CCCN(C(=O)O)C1

nearest known ligand 0.46

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.46
RAB9A P51151 1/20 0.46
KDM2B Q8NHM5 4/20 0.43
ALDH1A1 P00352 5/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
MAPT P10636 2/20 0.42
MAPK1 P28482 1/20 0.42
POLB P06746 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1869732 0.86 ALOX5AP (0.47) GAARAB9AKDM2BALDH1A1MEN1
SCHEMBL1869734 0.86 ALOX5AP (0.47) GAARAB9AKDM2BALDH1A1MEN1
SCHEMBL5593253 0.83 KDM2B (0.43) GAARAB9AKDM2BALDH1A1MEN1
SCHEMBL4982747 0.81 HPGD (0.54) GAARAB9AALDH1A1MEN1KMT2A
SCHEMBL2845267 0.78 GAA (0.45) GAARAB9AALDH1A1MEN1KMT2A
SCHEMBL4755206 0.77 POLB (0.52) GAARAB9AKDM2BALDH1A1MEN1
SCHEMBL4972616 0.74 ALDH1A1 (0.49) GAAKDM2BALDH1A1MEN1KMT2A
SCHEMBL23835159 0.72 PARP10 (0.52)
SCHEMBL5593568 0.72 RBP4 (0.41) RAB9AALDH1A1MEN1KMT2AMAPT
SCHEMBL5509718 0.70 REN (0.56)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101072561-B Diaminoalkane aspartic protease inhibitors VITAE PHARMACEUTICALS INC 2011-05-11 CN disclosed
CN-101072561-A Diaminoalkane aspartic protease inhibitors VITAE PHARMACEUTICALS INC (US) 2007-11-14 CN disclosed
EP-1807078-A1 DIAMINOALKANE ASPARTIC PROTEASE INHIBITORS Vitae Pharmaceuticals, Inc. (US) 2007-07-18 EP disclosed
WO-2006042150-A1 DIAMINOALKANE ASPARTIC PROTEASE INHIBITORS VITAE PHARMACEUTICALS, INC. (US) 2006-04-20 WO disclosed