SCHEMBL5511934

SCHEMBL5511934

COc1ccc2nccc(NC(=O)CCC3CCCNC3)c2n1

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.46
KCNH2 Q12809 4/20 0.43
ACP1 P24666 2/20 0.42
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.40
NPSR1 Q6W5P4 1/20 0.39
BRD4 O60885 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KDM1A O60341 1/20 0.39
PI4KB Q9UBF8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5512410 0.83 KCNH2 (0.44) KCNH2CNR1CNR2
SCHEMBL5509547 0.78 CYP2C9 (0.45) KCNH2KMT2AMEN1KDM4EALDH1A1
SCHEMBL590586 0.76 KCNH2 (0.46) KCNH2CNR1CNR2ALDH1A1NPC1
SCHEMBL5508579 0.75 ALDH1A1 (0.47) CNR1CNR2KMT2AMEN1ALDH1A1
SCHEMBL5508574 0.75 ALDH1A1 (0.47) CNR1CNR2KMT2AMEN1ALDH1A1
SCHEMBL633958 0.75 KCNH2 (0.54) KCNH2CNR1CNR2ALDH1A1
SCHEMBL591768 0.74 KDM4E (0.51) KCNH2KMT2AMEN1KDM4EALDH1A1
SCHEMBL5506636 0.73 KCNH2 (0.56) KCNH2KMT2AKDM4E
SCHEMBL5507933 0.73 KCNH2 (0.45) KCNH2CNR1CNR2KMT2AMEN1
SCHEMBL632652 0.72 KCNH2 (0.39) KCNH2CNR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799676-A2 NEW BICYCLIC ANTIBIOTICS Actelion Pharmaceuticals Ltd. (CH) 2007-06-27 EP disclosed
WO-2006032466-A2 NEW BICYCLIC ANTIBIOTICS ACTELION PHARMACEUTICALS LTD (CH) 2006-03-30 WO disclosed