Isatin

Isatin

SCHEMBL5510399

O=C1C(=O)N(CCF)c2ccccc21.O=C1Nc2ccccc2C1=O

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CES1 P23141 6/20 0.58
BCHE P06276 2/20 0.58
MAOA P21397 2/20 0.54
MAOB P27338 2/20 0.54
ALDH1A1 P00352 6/20 0.52
ALDH2 P05091 4/20 0.52
ALDH3A1 P30838 4/20 0.52
CDC25A P30304 1/20 0.51
PKM P14618 1/20 0.51
TP53 P04637 1/20 0.50
PARK7 Q99497 1/20 0.50
TGM2 P21980 1/20 0.50
PTPN1 P18031 1/20 0.48
HDAC8 Q9BY41 1/20 0.46
CHRM1 P11229 1/20 0.46
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5999219 0.85 CES1 (0.79) CES1BCHEMAOAMAOBALDH1A1
Isatin SCHEMBL5505028 0.83 MAOA (0.57) CES1BCHEMAOAMAOBALDH1A1
Isatin SCHEMBL25225927 0.80 MAOA (0.74) CES1BCHEMAOAMAOBALDH1A1
Isatin SCHEMBL9390159 0.77 ALDH3A1 (0.65) CES1BCHEALDH1A1ALDH3A1TP53
SCHEMBL25119569 0.76 CES1 (0.85) CES1BCHEMAOAMAOBALDH1A1
SCHEMBL19924204 0.75 CES1 (1.00) CES1BCHEMAOAMAOBALDH1A1
Isatin SCHEMBL5506077 0.75 MAOA (0.50) CES1BCHEMAOAMAOBALDH1A1
SCHEMBL25119255 0.74 CES1 (0.84) CES1BCHEMAOAMAOBALDH1A1
Isatin SCHEMBL34016 0.73 MAOA (1.00) CES1MAOAMAOBALDH1A1PKM
Isatin SCHEMBL973760 0.73 MAOA (1.00) CES1MAOAMAOBALDH1A1PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781642-A1 OXAZOLIDINONES CONTAINING OXINDOLES AS ANTIBACTERIAL AGENTS Pharmacia & Upjohn Company LLC (US) 2007-05-09 EP disclosed
WO-2006016221-A1 OXAZOLIDINONES CONTAINING OXINDOLES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-02-16 WO disclosed