SCHEMBL5511796

SCHEMBL5511796

CS(=O)(=O)Nc1ccc(I)cc1F.Nc1ccc(I)cc1F

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAP2K1 Q02750 1/20 0.41
CA1 P00915 2/20 0.40
CA2 P00918 2/20 0.40
CA12 O43570 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
CA5A P35218 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CA5B Q9Y2D0 1/20 0.40
LMNA P02545 1/20 0.40
FFAR4 Q5NUL3 1/20 0.39
KIT P10721 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1542413 0.91 MAP2K1 (0.43) MAP2K1
SCHEMBL2206288 0.77 LMNA (0.45) LMNAKIT
SCHEMBL26386555 0.77 KDM1A (0.48)
SCHEMBL188879 0.76
SCHEMBL392027 0.75 MAP2K1 (0.58) MAP2K1CA2
SCHEMBL18897008 0.75 ADRB3 (0.36) LMNA
SCHEMBL9464838 0.74 PSIP1 (0.59) MAP2K1LMNA
SCHEMBL18332099 0.74 KDM1A (0.40) CA1CA2CA9LMNAKIT
SCHEMBL10626704 0.73 PTGS2 (0.56) LMNAKIT
SCHEMBL27183049 0.72 CA2 (0.43) MAP2K1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1861358-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME Amorepacific Corporation (KR) 2007-12-05 EP disclosed
WO-2006101321-A1 NOVEL COMPOUNDS, ISOMER THEREOF, OR PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF AS VANILLOID RECEPTOR ANTAGONIST; AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AMOREPACIFIC CORPORATION (KR) 2006-09-28 WO disclosed