SCHEMBL5527952

SCHEMBL5527952

CCCc1nc(C#N)cn1CC(C)C

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
RPS6KB1 P23443 1/20 0.48
TLR7 Q9NYK1 1/20 0.32
PDE10A Q9Y233 2/20 0.32
CYP19A1 P11511 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
MAPT P10636 2/20 0.30
ALDH1A1 P00352 1/20 0.30
LMNA P02545 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
CTSS P25774 1/20 0.30
CTSK P43235 1/20 0.30
KDM4E B2RXH2 1/20 0.30
MEN1 O00255 1/20 0.30
THRB P10828 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27306641 0.75 CTSK (0.36) PDE10ACYP19A1MAPTALDH1A1LMNA
SCHEMBL5357748 0.65 RPS6KB1 (1.00) RPS6KB1
SCHEMBL10147185 0.65 KCNH2 (0.45) ALDH1A1KMT2A
SCHEMBL1301797 0.65 TLR7 (0.36) TLR7PDE10AMAPTALDH1A1LMNA
SCHEMBL1300750 0.65 TLR7 (0.41) RPS6KB1TLR7PDE10AMAPTALDH1A1
SCHEMBL17835018 0.64 BRD4 (0.33) RPS6KB1
SCHEMBL12881774 0.61 ALDH1A1 (0.31) MAPTALDH1A1LMNASMN1; SMN2
SCHEMBL5533170 0.61 RPS6KB1 (0.38) RPS6KB1HRH3MAPTKDM4EMEN1
SCHEMBL2066236 0.58 PDE10A (0.38) PDE10ACYP19A1CTSSCTSKKDM4E
SCHEMBL25291538 0.58 RPS6KB1 (0.38) RPS6KB1CYP19A1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1863770-A2 RING CLOSING AND RELATED METHODS AND INTERMEDIATES Coley Pharmaceutical Group, Inc. (US) 2007-12-12 EP disclosed
WO-2006121528-A2 RING CLOSING AND RELATED METHODS AND INTERMEDIATES COLEY PHARMACEUTICAL GROUP, INC. (US) 2006-11-16 WO disclosed