SCHEMBL5530790

SCHEMBL5530790

O=C(Nc1ccccn1)C(=O)c1c(Cc2ccc(F)cc2)[nH]c2ccccc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.43
PKM P14618 2/20 0.43
RAB9A P51151 2/20 0.43
GABRP O00591 1/20 0.41
GABRD O14764 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRB2 P47870 1/20 0.41
GABRA4 P48169 1/20 0.41
GABRE P78334 1/20 0.41
GABRA6 Q16445 1/20 0.41
GABRG1 Q8N1C3 1/20 0.41
GABRG3 Q99928 1/20 0.41
GABRQ Q9UN88 1/20 0.41
DHODH Q02127 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5533387 0.91 NPC1 (0.47) NPC1PKMRAB9AMEN1KMT2A
SCHEMBL5531131 0.85 RAB9A (0.47) NPC1RAB9AGABRPGABRDGABRA1
SCHEMBL5535174 0.85 MAPT (0.46) NPC1RAB9AGABRPGABRDGABRA1
SCHEMBL5535769 0.84 GABRP (0.42) NPC1RAB9AGABRPGABRDGABRA1
SCHEMBL5532784 0.82 PDE4A (0.52) NPC1PKMRAB9AMEN1KMT2A
SCHEMBL8804285 0.81 KMT2A (0.47) NPC1RAB9ADHODHVDRMEN1
SCHEMBL5528849 0.81 MEN1 (0.42) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL5528306 0.78 KMT2A (0.47) MEN1KMT2AGAA
SCHEMBL5538626 0.77 MAPT (0.57) NPC1RAB9AMEN1KMT2ASMN1; SMN2
SCHEMBL4029345 0.75 POLB (0.45) NPC1RAB9AMEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1809279-A1 NANOPARTICULATE COMPOSITIONS OF TUBULIN INHIBITOR BAXTER INTERNATIONAL INC. (US) 2007-07-25 EP claimed
WO-2006052712-A1 NANOPARTICULATE COMPOSITIONS OF TUBULIN INHIBITOR BAXTER INTERNATIONAL INC. (US) 2006-05-18 WO claimed