SCHEMBL5533938

SCHEMBL5533938

CN1C=CN(c2cc(F)ccc2C#N)N1

nearest known ligand 0.35

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.34
FFAR4 Q5NUL3 1/20 0.34
CYP11B1 P15538 3/20 0.33
CYP11B2 P19099 3/20 0.33
AR P10275 3/20 0.33
GABRA1 P14867 3/20 0.31
GABRG2 P18507 3/20 0.31
GABRB3 P28472 3/20 0.31
GABRA5 P31644 3/20 0.31
GABRA3 P34903 3/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
PGR P06401 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Iodide SCHEMBL27085270 0.79 L3MBTL1 (0.35)
SCHEMBL19812737 0.73 KDM4E (0.50)
SCHEMBL29817937 0.69 ALDH1A1 (0.55) FFAR4
SCHEMBL2520368 0.68 MAPT (0.41)
SCHEMBL2528786 0.67 GABRA1 (0.42) FFAR4CYP11B2ARGABRA1GABRG2
SCHEMBL57346 0.66 TRPV4 (0.61) TRPV4CYP11B1CYP11B2ARMAOA
SCHEMBL30919072 0.66 TRPV4 (0.61) TRPV4CYP11B1CYP11B2ARMAOA
SCHEMBL2526428 0.66 CDK4 (0.38) FFAR4ARPGR
SCHEMBL2523972 0.66 HCRTR2 (0.39) TRPV4FFAR4CYP11B1CYP11B2MAOA
SCHEMBL17871934 0.66 AR (0.51) FFAR4CYP11B1CYP11B2AR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1749011-A1 BICYCLIC HETEROCYCLES AS HIV INTEGRASE INHIBITORS Bristol-Myers Squibb Company (US) 2007-02-07 EP disclosed
WO-2005118593-A1 BICYCLIC HETEROCYCLES AS HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2005-12-15 WO disclosed