SCHEMBL5534487

SCHEMBL5534487

CCn1c(C2(OCCO)CCN(C(=O)OCc3ccccc3)C2)nc(C(=O)O)c(O)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACB O00763 1/20 0.39
ENPP2 Q13822 1/20 0.39
ATXN2 Q99700 1/20 0.39
ADORA2B P29275 1/20 0.37
OPRD1 P41143 2/20 0.36
OPRK1 P41145 2/20 0.36
RORC P51449 3/20 0.36
HDAC1 Q13547 3/20 0.36
HDAC6 Q9UBN7 3/20 0.36
HDAC3 O15379 2/20 0.36
HDAC2 Q92769 2/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
MKNK1 Q9BUB5 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
FNTA P49354 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5528302 0.95 ENPP2 (0.40) ACACBENPP2ATXN2ADORA2BOPRD1
SCHEMBL5538682 0.90 ADORA2B (0.40) ACACBENPP2ATXN2ADORA2BOPRD1
SCHEMBL5527354 0.81 OPRK1 (0.39) ACACBENPP2ATXN2ADORA2BOPRD1
SCHEMBL5532804 0.79 HDAC1 (0.43) ACACBENPP2ATXN2ADORA2BOPRD1
SCHEMBL5534382 0.79 OPRD1 (0.40) ACACBENPP2ATXN2ADORA2BOPRD1
SCHEMBL2083125 0.76 ACACB (0.43) ACACBENPP2ATXN2ADORA2BOPRD1
SCHEMBL5536389 0.74 ENPP2 (0.36) ACACBENPP2ATXN2ADORA2BOPRD1
SCHEMBL2081516 0.73 ENPP2 (0.43) ACACBENPP2ATXN2ADORA2BOPRD1
SCHEMBL1117837 0.71 CTSB (0.36) SMN1; SMN2
SCHEMBL9901321 0.70 SMN1; SMN2 (0.35) RORCMEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007143446-A1 SPIRO-CONDENSED HETEROTRICYCLIC COMPOUNDS AS HIV INTEGRASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2007-12-13 WO disclosed