SCHEMBL5540347

SCHEMBL5540347

CC(C)(C)c1ccc(C(=O)NC2N=CC3=CN(S(=O)(=O)c4ccccc4F)CCC3=N2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCKAR P32238 2/20 0.39
CCKBR P32239 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
KMT2A Q03164 5/20 0.38
MEN1 O00255 2/20 0.38
EPHX2 P34913 1/20 0.35
ALDH1A1 P00352 3/20 0.34
STAT3 P40763 2/20 0.33
TRPV1 Q8NER1 1/20 0.33
HSD11B1 P28845 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
TSHR P16473 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAB9A P51151 1/20 0.33
PTGER2 P43116 2/20 0.33
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5548484 0.76 KMT2A (0.54) KMT2AMEN1ALDH1A1RAB9A
SCHEMBL5540364 0.75 CPT2 (0.39) L3MBTL1KMT2AMEN1MAPK1SMN1; SMN2
SCHEMBL5540355 0.74 CA1 (0.39) L3MBTL1KMT2AALDH1A1TRPV1HSD11B1
SCHEMBL5546851 0.72 KMT2A (0.39) L3MBTL1KMT2AMEN1CYP2D6CYP2C19
SCHEMBL5546858 0.72 MEN1 (0.38) KMT2AMEN1EPHX2ALDH1A1CYP2D6
SCHEMBL5545022 0.72 MEN1 (0.36) KMT2AMEN1ALDH1A1RAB9ASMN1; SMN2
SCHEMBL5546920 0.71 HTR3E (0.39) KMT2AMEN1RAB9ASMN1; SMN2
SCHEMBL5546197 0.66 NOD2 (0.39) KMT2AMEN1ALDH1A1SMN1; SMN2
SCHEMBL5540335 0.66 PGR (0.36) L3MBTL1KMT2AALDH1A1HSD11B1
SCHEMBL5546694 0.63 HTR3A (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed