SCHEMBL5540335

SCHEMBL5540335

O=C(NC1N=CC2=CN(C(=O)c3ccc(Cl)c(Cl)c3)CCC2=N1)c1ccccc1F

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PGR P06401 3/20 0.36
GPR6 P46095 1/20 0.36
GRM5 P41594 1/20 0.35
ALDH1A1 P00352 2/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
KMT2A Q03164 2/20 0.34
HPGD P15428 1/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNA7 P36544 1/20 0.33
CHRNA4 P43681 1/20 0.33
GRM4 Q14833 1/20 0.33
HSD11B1 P28845 1/20 0.33
CCR3 P51677 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5540342 0.74 ALDH1A1 (0.39) PGRALDH1A1L3MBTL1KMT2AHPGD
SCHEMBL5544982 0.72 HPGDS (0.42)
SCHEMBL5546833 0.70 FLT1 (0.42) PGRALDH1A1KMT2ACHRNA7
SCHEMBL5546196 0.67 TRPV1 (0.38) GPR6
SCHEMBL5546568 0.66 CHRM1 (0.38) KMT2A
SCHEMBL5544998 0.66 SIGMAR1 (0.41)
SCHEMBL5546606 0.64 OPRK1 (0.35) ALDH1A1KMT2AHPGD
SCHEMBL5540386 0.64 LMNA (0.34) ALDH1A1KMT2A
SCHEMBL5548485 0.63 KMT2A (0.37) KMT2A
SCHEMBL5540365 0.62 KMT2A (0.36) ALDH1A1KMT2ACHRNA7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed