SCHEMBL5540374

SCHEMBL5540374

O=C(NC1=NCC2=CN(C(=O)c3cc(F)cc4c3OCOC4)CCC2=N1)c1ccccc1C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CXCR5 P32302 1/20 0.38
PTGES O14684 5/20 0.37
KDM4E B2RXH2 2/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CNR1 P21554 4/20 0.34
CNR2 P34972 4/20 0.34
TP53 P04637 2/20 0.33
LMNA P02545 1/20 0.33
POLB P06746 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
GALR3 O60755 1/20 0.32
NR2F2 P24468 1/20 0.32
MAPK8 P45983 1/20 0.32
F11 P03951 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545032 0.76 PTGES (0.39) PTGESTP53LMNA
SCHEMBL5537975 0.75 RXFP1 (0.39) PTGESTP53LMNA
SCHEMBL5538007 0.74 PTGES (0.39) PTGESCNR1CNR2TP53LMNA
SCHEMBL3527453 0.71 KDR (0.41) CXCR5PTGESKDM4ENPC1RAB9A
SCHEMBL5548741 0.66 SMN1; SMN2 (0.41) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL5546600 0.66 KMT2A (0.40) KDM4ENPC1RAB9AALDH1A1TP53
SCHEMBL5538068 0.65 MAPT (0.39) KDM4ENPC1RAB9AKMT2A
SCHEMBL5538119 0.64 RAB9A (0.46) NPC1RAB9AALDH1A1TP53LMNA
SCHEMBL5540369 0.63 CPT2 (0.40) KDM4EALDH1A1TP53LMNAMEN1
SCHEMBL5546603 0.62 HPGDS (0.39) KDM4ENPC1RAB9AALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed