SCHEMBL5546600

SCHEMBL5546600

O=C(NC1=NCC2=CN(C(=O)c3ccc(F)cc3)CCC2=N1)c1cccc(F)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.40
MEN1 O00255 3/20 0.40
SMN1; SMN2 Q16637 5/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
TSHR P16473 3/20 0.39
MAPT P10636 3/20 0.39
TP53 P04637 2/20 0.39
KDM4E B2RXH2 2/20 0.39
KCNQ3 O43525 2/20 0.39
KCNQ2 O43526 2/20 0.39
KCNQ5 Q9NR82 1/20 0.39
ALDH1A1 P00352 1/20 0.38
GLA P06280 1/20 0.38
PKM P14618 1/20 0.38
ADCY1 Q08828 1/20 0.38
MAPK1 P28482 1/20 0.38
KCNE1 P15382 1/20 0.38
KCNQ1 P51787 1/20 0.38
NFKB1 P19838 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5548741 0.84 SMN1; SMN2 (0.41) KMT2AMEN1SMN1; SMN2NPC1RAB9A
SCHEMBL5548146 0.82 MAPT (0.48) KMT2AMEN1SMN1; SMN2RAB9AMAPT
SCHEMBL5544949 0.80 ALDH1A1 (0.36) KMT2AMEN1SMN1; SMN2NPC1RAB9A
SCHEMBL5546854 0.80 CYP2C19 (0.40) KMT2AMEN1SMN1; SMN2NPC1RAB9A
SCHEMBL5546603 0.80 HPGDS (0.39) KMT2AMEN1SMN1; SMN2NPC1RAB9A
SCHEMBL5540828 0.77 MAPT (0.44) KMT2AMEN1MAPTKDM4EALDH1A1
SCHEMBL5538119 0.76 RAB9A (0.46) KMT2AMEN1SMN1; SMN2NPC1RAB9A
SCHEMBL5545053 0.76 GRM5 (0.39) KMT2AMEN1NPC1RAB9AMAPT
SCHEMBL5546202 0.75 NOD2 (0.40) KMT2AMEN1SMN1; SMN2NPC1RAB9A
SCHEMBL5543044 0.75 MGLL (0.38) KMT2AMEN1SMN1; SMN2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed