SCHEMBL5538007

SCHEMBL5538007

O=C(NC1=NCC2=CN(C(=O)C3CCCCC3)CCC2=N1)c1ccccc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PTGES O14684 8/20 0.39
TP53 P04637 1/20 0.38
RXFP1 Q9HBX9 4/20 0.37
HCRTR1 O43613 1/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
PTGS1 P23219 1/20 0.35
ACKR3 P25106 1/20 0.35
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545032 0.83 PTGES (0.39) PTGESTP53PTGS1ACKR3LMNA
SCHEMBL5546183 0.79 GRM5 (0.44) PTGESTP53PTGS1LMNAGAA
SCHEMBL5537975 0.77 RXFP1 (0.39) PTGESTP53RXFP1PTGS1LMNA
SCHEMBL5540374 0.74 CXCR5 (0.38) PTGESTP53CNR1CNR2LMNA
SCHEMBL5538002 0.74 HCRTR1 (0.40) PTGESTP53HCRTR1LMNAGAA
SCHEMBL5546875 0.67 MAPT (0.38) TP53HCRTR1CNR1CNR2LMNA
SCHEMBL5546353 0.66 KEAP1 (0.47) PTGES
SCHEMBL5546883 0.64 KDM4E (0.40) TP53RXFP1HCRTR1LMNAGAA
SCHEMBL5546600 0.62 KMT2A (0.40) TP53LMNA
SCHEMBL6930440 0.62 LMNA (0.63) PTGESLMNAGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed