SCHEMBL5543044

SCHEMBL5543044

O=C(NC1=NCC2=CN(C(=O)c3ccc(OC(F)(F)F)cc3)CCC2=N1)c1cc(Cl)cc(Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 1/20 0.38
TRPV1 Q8NER1 2/20 0.37
ABL1 P00519 6/20 0.36
EPHX2 P34913 3/20 0.36
TNF P01375 1/20 0.35
NOD2 Q9HC29 1/20 0.35
NOD1 Q9Y239 1/20 0.35
GCGR P47871 2/20 0.35
GIPR P48546 2/20 0.35
MEN1 O00255 1/20 0.35
HTT P42858 1/20 0.35
KMT2A Q03164 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
KCNK2 O95069 1/20 0.35
KCNK10 P57789 1/20 0.35
RAPGEF3 O95398 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5546201 0.77 ABL1 (0.40) TRPV1ABL1EPHX2MEN1HTT
SCHEMBL5546600 0.75 KMT2A (0.40) MEN1HTTKMT2ASMN1; SMN2
SCHEMBL5543042 0.73 MGLL (0.39) MGLLTRPV1EPHX2GCGRGIPR
SCHEMBL5546875 0.72 MAPT (0.38) MEN1HTTKMT2ASMN1; SMN2
SCHEMBL5544987 0.71 PRKAA2 (0.42)
SCHEMBL5546870 0.68 NAMPT (0.34) EPHX2HTTKMT2ASMN1; SMN2
SCHEMBL5538119 0.67 RAB9A (0.46) MEN1HTTKMT2ASMN1; SMN2
SCHEMBL5537975 0.66 RXFP1 (0.39)
SCHEMBL5545017 0.66 ALDH1A1 (0.41) MEN1KMT2ASMN1; SMN2
SCHEMBL5548490 0.66 MAPT (0.39) MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed