SCHEMBL5544746

SCHEMBL5544746

CC(C)(C)OC(=O)C(CCN1C(=O)c2ccccc2C1=O)O[Si](C)(C)C

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.41
ALDH1A1 P00352 5/20 0.41
LMNA P02545 1/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
GAA P10253 1/20 0.39
TP53 P04637 1/20 0.39
PKM P14618 1/20 0.39
HPGD P15428 1/20 0.39
MAPT P10636 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
GLA P06280 1/20 0.38
BRCA1 P38398 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6291909 0.82 PKM (0.47) SMN1; SMN2ALDH1A1GAAPKMHPGD
SCHEMBL13384515 0.81 ALDH1A1 (0.47) SMN1; SMN2ALDH1A1MEN1KMT2AGAA
SCHEMBL878178 0.80 SMN1; SMN2 (0.45) SMN1; SMN2ALDH1A1GAAPKMMMP2
SCHEMBL18918957 0.77 MMP2 (0.46) SMN1; SMN2MEN1KMT2APKMMAPT
SCHEMBL442293 0.75 MMP2 (0.44) SMN1; SMN2ALDH1A1LMNAMEN1KMT2A
SCHEMBL5031610 0.75 MMP2 (0.44) SMN1; SMN2MEN1KMT2AMAPTMMP2
SCHEMBL9322023 0.74 HDAC1 (0.47) SMN1; SMN2ALDH1A1LMNAMEN1KMT2A
SCHEMBL15887315 0.74 PKM (0.36) ALDH1A1MEN1KMT2ATP53PKM
SCHEMBL10215923 0.73 ALDH1A1 (0.48) ALDH1A1PKMHPGDMAPTNPSR1
SCHEMBL22559290 0.72 AKT1 (0.43) ALDH1A1MEN1KMT2ATP53PKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1799653-B1 Condensed thienopyrimidine derivatives for the treatment of cancer BAYER IP GMBH (DE) 2013-03-20 EP disclosed
EP-1799653-A2 NOVEL HETEROCYCLES Bayer Pharmaceuticals Corporation (US) 2007-06-27 EP disclosed
WO-2006023843-A2 NOVEL HETEROCYCLES BAYER PHARMACEUTICALS CORPORATION (US) 2006-03-02 WO disclosed