SCHEMBL5544982

SCHEMBL5544982

O=C(NC1N=CC2=CN(C(=O)c3ccc(Oc4ccccc4)nc3)CCC2=N1)c1ccc(F)c(F)c1

nearest known ligand 0.42

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HPGDS O60760 1/20 0.42
PRKAA2 P54646 2/20 0.42
HRH3 Q9Y5N1 11/20 0.39
OPRM1 P35372 1/20 0.36
KCNH2 Q12809 1/20 0.36
MGLL Q99685 1/20 0.35
MCHR1 Q99705 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
DGAT1 O75907 1/20 0.35
SOAT1 P35610 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5546694 0.79 HTR3A (0.45) MGLLMCHR1
SCHEMBL5544987 0.76 PRKAA2 (0.42) HPGDSPRKAA2HRH3OPRM1DGAT1
SCHEMBL3533032 0.67 PDGFRB (0.49) PRKAA2HRH3
SCHEMBL5546197 0.67 NOD2 (0.39) HRH3MCHR1SMN1; SMN2
SCHEMBL5544998 0.65 SIGMAR1 (0.41) HRH3KCNH2MCHR1
SCHEMBL5546858 0.65 MEN1 (0.38) SMN1; SMN2
SCHEMBL5546920 0.64 HTR3E (0.39) HPGDSSMN1; SMN2
SCHEMBL5546568 0.64 CHRM1 (0.38) PRKAA2HRH3
SCHEMBL6179704 0.62 KCNQ3 (0.58) PRKAA2DGAT1SOAT1
SCHEMBL5540386 0.62 LMNA (0.34) OPRM1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed