SCHEMBL5546162

SCHEMBL5546162

CCCCC(C)CCC(=O)N1C=C2C=NC(NC(=O)c3ccc(F)cc3)N=C2CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
GAA P10253 1/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
KDM5A P29375 1/20 0.32
SLC6A12 P48065 1/20 0.32
TMEM97 Q5BJF2 1/20 0.32
MCHR1 Q99705 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31
CHRNB2 P17787 1/20 0.31
CHRNA7 P36544 1/20 0.31
CHRNA4 P43681 1/20 0.31
OPRK1 P41145 1/20 0.31
CCR3 P51677 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CTSB P07858 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5540250 0.75 LMNA (0.39) SLC6A12TMEM97MCHR1SIGMAR1DRD2
SCHEMBL5546164 0.74 ALDH1A1 (0.34) ALDH1A1HPGDGAAHDAC3HDAC1
SCHEMBL5548143 0.73 MAPT (0.43) ALDH1A1GAASLC6A12TMEM97MCHR1
SCHEMBL5546932 0.72 TDP1 (0.36) ALDH1A1DRD2DRD4CHRNB2CHRNA7
SCHEMBL5546858 0.70 MEN1 (0.38) ALDH1A1HPGDSMN1; SMN2
SCHEMBL5546598 0.69 HPGDS (0.37) SIGMAR1DRD2DRD4CHRNB2CHRNA4
SCHEMBL15643184 0.67 F2 (0.40) MCHR1SIGMAR1DRD4CHRNB2CHRNA7
SCHEMBL5546891 0.67 KMT2A (0.39) ALDH1A1HPGDGAASMN1; SMN2LMNA
SCHEMBL5548484 0.67 KMT2A (0.54) ALDH1A1GAACCR3LMNA
SCHEMBL5546197 0.66 NOD2 (0.39) ALDH1A1HDAC3HDAC1HDAC2SLC6A12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed