SCHEMBL5546164

SCHEMBL5546164

CCCCC(C)CCC(=O)N1C=C2CN=C(NC(=O)c3ccc(F)cc3)N=C2CC1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.34
HPGD P15428 1/20 0.34
GAA P10253 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.32
RAB9A P51151 2/20 0.32
HDAC3 O15379 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC2 Q92769 1/20 0.32
CCR8 P51685 1/20 0.32
HTR1F P30939 2/20 0.32
ALOX15 P16050 1/20 0.31
CASP1 P29466 1/20 0.31
HSD17B10 Q99714 1/20 0.31
SAE1 Q9UBE0 1/20 0.31
UBA2 Q9UBT2 1/20 0.31
KMT2A Q03164 2/20 0.31
HTR7 P34969 1/20 0.31
KDM4E B2RXH2 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
KDM1A O60341 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5546162 0.74 ALDH1A1 (0.34) ALDH1A1HPGDGAASMN1; SMN2HDAC3
SCHEMBL3531277 0.67 CYP1A2 (0.42) ALDH1A1HTR1FKDM4E
SCHEMBL27460356 0.54 KMT2A (0.59) RAB9ACCR8KMT2A
SCHEMBL12706070 0.54 ALDH1A1 (1.00) ALDH1A1HPGDSMN1; SMN2RAB9AHDAC3
SCHEMBL17474023 0.54 HDAC3 (0.57) ALDH1A1HPGDGAAHDAC3HDAC1
SCHEMBL28929300 0.53 GAA (0.73) ALDH1A1HPGDGAASMN1; SMN2HDAC3
SCHEMBL18086890 0.53 LMNA (0.44) ALDH1A1HPGDGAASMN1; SMN2RAB9A
SCHEMBL24386079 0.53 L3MBTL1 (0.71) ALDH1A1GAASMN1; SMN2RAB9AHDAC3
SCHEMBL16229517 0.53 ALDH1A1 (0.55) ALDH1A1HPGDSMN1; SMN2RAB9AHDAC3
SCHEMBL9665425 0.52 HTR7 (0.53) ALDH1A1HPGDGAASMN1; SMN2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed