SCHEMBL5546180

SCHEMBL5546180

O=C(NC1N=CC2=CN(C(=O)CN3C(=O)c4ccccc4C3=O)CCC2=N1)c1ccccc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SCN4A P35499 1/20 0.34
SCN9A Q15858 1/20 0.34
PPIA P62937 1/20 0.34
CYP2C9 P11712 2/20 0.33
CYP2C19 P33261 2/20 0.33
HTR2B P41595 1/20 0.33
MAPK14 Q16539 1/20 0.33
TP53 P04637 2/20 0.33
HCRTR1 O43613 1/20 0.33
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
LMNA P02545 1/20 0.32
GAA P10253 1/20 0.32
DPP4 P27487 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545030 0.86 CYP2C9 (0.36) SCN4ASCN9ACYP2C9CYP2C19HTR2B
SCHEMBL5538002 0.80 HCRTR1 (0.40) CYP2C9CYP2C19HTR2BMAPK14TP53
SCHEMBL5546183 0.74 GRM5 (0.44) GRM5MEN1KMT2ASMN1; SMN2CYP2C9
SCHEMBL5544998 0.72 SIGMAR1 (0.41) SCN9A
SCHEMBL5548485 0.65 KMT2A (0.37) MEN1KMT2ACYP2C19HCRTR1GAA
SCHEMBL5546460 0.63 MEN1 (0.43) GRM5MEN1KMT2ASMN1; SMN2KDM4E
SCHEMBL5546606 0.62 OPRK1 (0.35) MEN1KMT2ASMN1; SMN2CYP2C19KDM4E
SCHEMBL5540386 0.60 LMNA (0.34) MEN1KMT2ASMN1; SMN2ALDH1A1LMNA
SCHEMBL25239750 0.60 PTGS1 (0.63) GRM5MEN1KMT2AL3MBTL1PPIA
SCHEMBL1819622 0.58 LMNA (0.62) PPIATP53HCRTR1KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed