SCHEMBL5546183

SCHEMBL5546183

O=C(NC1=NCC2=CN(C(=O)CN3C(=O)c4ccccc4C3=O)CCC2=N1)c1ccccc1C(F)(F)F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.44
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
PTPRC P08575 1/20 0.36
TP53 P04637 1/20 0.36
RECQL P46063 1/20 0.34
PDE3B Q13370 1/20 0.33
PDE3A Q14432 1/20 0.33
PTGES O14684 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
GAA P10253 2/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
PTGS1 P23219 1/20 0.32
KCNK3 O14649 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545032 0.86 PTGES (0.39) GRM5TP53RECQLPDE3BPDE3A
SCHEMBL5538007 0.79 PTGES (0.39) TP53PTGESGAALMNAPTGS1
SCHEMBL5537975 0.75 RXFP1 (0.39) GRM5TP53PTGESCYP3A4CYP2C9
SCHEMBL5546180 0.74 GRM5 (0.40) GRM5MEN1KMT2APTPRCTP53
SCHEMBL5540374 0.72 CXCR5 (0.38) MEN1KMT2ATP53PTGESKDM4E
SCHEMBL5546883 0.68 KDM4E (0.40) MEN1KMT2ATP53KDM4EALDH1A1
SCHEMBL5546460 0.67 MEN1 (0.43) GRM5MEN1KMT2AKDM4EALDH1A1
SCHEMBL5546875 0.64 MAPT (0.38) MEN1KMT2ATP53ALDH1A1LMNA
SCHEMBL5546600 0.61 KMT2A (0.40) MEN1KMT2ATP53KDM4EALDH1A1
SCHEMBL25239750 0.61 PTGS1 (0.63) GRM5MEN1KMT2APTPRCRECQL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed