SCHEMBL5546895

SCHEMBL5546895

CCc1ccc(C(=O)NC2=NCC3=CN(C(=O)C4CCCO4)CCC3=N2)cc1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.40
RAB9A P51151 4/20 0.38
NPC1 O15118 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
ALDH1A1 P00352 4/20 0.38
MAPT P10636 2/20 0.37
ADCY1 Q08828 1/20 0.36
HPGD P15428 3/20 0.36
HTT P42858 1/20 0.36
POLB P06746 3/20 0.36
KDM4E B2RXH2 1/20 0.36
TP53 P04637 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
TSHR P16473 1/20 0.36
GAA P10253 1/20 0.35
TRPV1 Q8NER1 1/20 0.35
HSD17B10 Q99714 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5540390 0.79 RAB9A (0.35) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL5546861 0.71 NR1H4 (0.38) RAB9ANPC1SMN1; SMN2ALDH1A1MAPT
SCHEMBL3529902 0.67 PDGFRB (0.46) KMT2AMAPTPOLBKDM4ETP53
SCHEMBL5546870 0.66 NAMPT (0.34) KMT2ARAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL5546603 0.63 HPGDS (0.39) KMT2ARAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL5545017 0.60 ALDH1A1 (0.41) KMT2ARAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL8404658 0.60 KMT2A (0.81) KMT2ARAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL5548489 0.59 TUBB4A (0.50) KMT2ARAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL17078749 0.57 HDAC6 (0.51) KMT2ARAB9ANPC1SMN1; SMN2ALDH1A1
SCHEMBL20432728 0.57 HDAC6 (0.51) KMT2ARAB9ANPC1SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007534719-A 2007-11-29 JP claimed
EP-1742925-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2007-01-17 EP claimed
WO-2005105759-A1 SUBSTITUTED 5, 6, 7, 8-TETRAHYDRO-PYRIDO[4, 3-D]PYRIMIDINE-2-YL COMPOUNDS AND 5, 6, 7, 8-TETRAHYDRO-QUINAZOLINE-2-YL COMPOUNDS Grünenthal GmbH (DE) 2005-11-10 WO claimed