SCHEMBL5548613

SCHEMBL5548613

COc1ccc(CCC(C)Nc2nc(C(C)(C)C)cn3c(=O)[nH]nc23)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 4/20 0.41
MAPK1 P28482 3/20 0.41
MAPT P10636 4/20 0.40
MEN1 O00255 2/20 0.40
POLB P06746 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 2/20 0.40
GSK3A P49840 3/20 0.39
GSK3B P49841 3/20 0.39
HTT P42858 2/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALDH1A1 P00352 4/20 0.39
GAA P10253 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
NPC1 O15118 1/20 0.35
G6PD P11413 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5545429 0.84 GSK3B (0.46) MAPTGSK3AGSK3B
SCHEMBL5550039 0.83 GSK3A (0.46) MAPTMEN1POLBKMT2AGSK3A
SCHEMBL3522851 0.78 CXCR2 (0.35)
SCHEMBL5548540 0.77 PDE5A (0.32) L3MBTL1MAPTKDM4EGSK3AGSK3B
SCHEMBL3529920 0.77 GSK3A (0.61) L3MBTL1MEN1KMT2AKDM4EGSK3A
SCHEMBL5549261 0.73 KMT2A (0.48) MAPK1MAPTMEN1POLBKMT2A
SCHEMBL5543524 0.72 ADORA1 (0.43) GSK3AGSK3B
SCHEMBL5543493 0.72 GSK3B (0.50) MAPTGSK3AGSK3BSMN1; SMN2
SCHEMBL5549402 0.72 ADORA1 (0.43) MAPTMEN1KMT2AGSK3AGSK3B
SCHEMBL5548609 0.72 MAPK1 (0.37) MAPK1MEN1KMT2AGSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed