SCHEMBL5550102

SCHEMBL5550102

CN(CCCNc1nc(C(C)(C)C)cn2c(=O)[nH]nc12)C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCNE2 O96020 1/20 0.35
CCNE1 P24864 1/20 0.35
CDK2 P24941 1/20 0.35
METAP2 P50579 1/20 0.34
BRD4 O60885 9/20 0.33
GSK3A P49840 7/20 0.32
GSK3B P49841 7/20 0.32
AAK1 Q2M2I8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3529268 0.80 ADORA1 (0.37) GSK3AGSK3B
SCHEMBL5549838 0.73 PGK1 (0.40) GSK3AGSK3B
SCHEMBL5543567 0.73 ADORA1 (0.47) GSK3AGSK3B
SCHEMBL3528788 0.73 GSK3B (0.34) GSK3AGSK3B
SCHEMBL3524574 0.72 GSK3B (0.32) GSK3AGSK3B
SCHEMBL5545429 0.71 GSK3B (0.46) GSK3AGSK3B
SCHEMBL4072562 0.70 AAK1 (0.38) CCNE2CCNE1CDK2METAP2BRD4
SCHEMBL5548616 0.70 CA12 (0.40) GSK3AGSK3B
SCHEMBL5549261 0.69 KMT2A (0.48)
SCHEMBL3526413 0.69 PKM (0.42) GSK3AGSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1678180-B1 SUBSTITUTED 2H-[1,2,4]TRIAZOLO 4,3-A PYRAZINES AS GSK-3 INHIBITORS PFIZER PROD INC (US) 2007-08-08 EP disclosed