SCHEMBL5552417

SCHEMBL5552417

CCOC(=O)Cc1nc(I)sc1C(=O)OCC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
HSD17B10 Q99714 3/20 0.46
CYP1A2 P05177 1/20 0.44
MC4R P32245 1/20 0.42
HPGD P15428 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 2/20 0.40
PPARG P37231 1/20 0.40
NCOA2 Q15596 1/20 0.40
RXFP1 Q9HBX9 1/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
TSHR P16473 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
CDC7 O00311 3/20 0.39
DBF4 Q9UBU7 3/20 0.39
TRPM8 Q7Z2W7 2/20 0.39
GAA P10253 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2719635 0.84 NPC1 (0.49) ALDH1A1HSD17B10CYP1A2MC4RHPGD
SCHEMBL30740576 0.83 ALDH1A1 (0.47) ALDH1A1HSD17B10CYP1A2HPGDLMNA
SCHEMBL2720641 0.82 ALDH1A1 (0.63) ALDH1A1HSD17B10CYP1A2HPGDLMNA
SCHEMBL15581984 0.82 ALDH1A1 (0.46) ALDH1A1HSD17B10CYP1A2HPGDLMNA
SCHEMBL2720481 0.82 ALDH1A1 (0.46) ALDH1A1HSD17B10CYP1A2MC4RHPGD
SCHEMBL2717529 0.79 LMNA (0.63) ALDH1A1HSD17B10CYP1A2HPGDLMNA
SCHEMBL3454027 0.79 ALDH1A1 (0.58) ALDH1A1HSD17B10CYP1A2HPGDLMNA
SCHEMBL3332542 0.78 ALDH1A1 (0.66) ALDH1A1HSD17B10CYP1A2MC4RHPGD
SCHEMBL26288487 0.76 ALDH1A1 (0.47) ALDH1A1HSD17B10CYP1A2MC4RHPGD
SCHEMBL2582135 0.75 TRPM8 (0.68) ALDH1A1HSD17B10MAPTSMN1; SMN2CDC7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012059041-A1 NOVEL 6-ARYLAMINO PYRIDONE CARBOXAMIDE AS MEK INHIBITORS CENTAURUS BIOPHARMA CO., LTD. (CN) 2012-05-10 WO disclosed