SCHEMBL5554008

SCHEMBL5554008

C[C@H](c1ccc(-c2ccc(-c3ccc(Cl)c(Cl)c3)cc2)cc1)N1CCCC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 8/20 0.48
SLC6A2 P23975 7/20 0.48
SLC6A4 P31645 7/20 0.48
AHR P35869 2/20 0.47
CYP2D6 P10635 2/20 0.43
CYP1B1 Q16678 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
HPGD P15428 1/20 0.41
PTGS1 P23219 1/20 0.40
ALDH1A1 P00352 1/20 0.40
GAA P10253 1/20 0.40
ADAM17 P78536 1/20 0.40
MCL1 Q07820 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
OPRK1 P41145 2/20 0.40
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
CYP3A4 P08684 1/20 0.39
UTS2R Q9UKP6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447344 1.00 SLC6A3 (0.48) SLC6A3SLC6A2SLC6A4AHRCYP2D6
SCHEMBL31669101 0.88 SLC6A3 (0.55) SLC6A3SLC6A2SLC6A4CYP2D6MEN1
SCHEMBL22206745 0.86 SLC6A3 (0.56) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL22206766 0.86 SLC6A3 (0.56) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL29585835 0.86 SLC6A3 (0.56) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL29585404 0.86 SLC6A3 (0.56) SLC6A3SLC6A2SLC6A4MEN1KMT2A
SCHEMBL6447211 0.86 CYP2D6 (0.40) SLC6A3SLC6A2SLC6A4CYP2D6CHRM2
SCHEMBL11626449 0.86 SLC6A2 (0.51) SLC6A3SLC6A2SLC6A4AHRCYP2D6
SCHEMBL5555138 0.83 CYP2D6 (0.43) SLC6A3SLC6A2SLC6A4CYP2D6ALDH1A1
SCHEMBL11623680 0.81 OGA (0.46) MEN1KMT2AALDH1A1SMN1; SMN2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1756058-A1 HISTAMINE-3 RECEPTOR ANTAGONISTS Pfizer Products Incorporated (US) 2007-02-28 EP disclosed
WO-2005105744-A1 HISTAMINE-3 RECEPTOR ANTAGONISTS PFIZER PRODUCTS INC. 2005-11-10 WO disclosed