SCHEMBL5558706

SCHEMBL5558706

CC[C@@H](C)c1c(OC)c(F)cc2c1c(OC(C)=O)c(C)n2C(=O)c1ccc(OC(F)F)cc1

nearest known ligand 0.37

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PPARG P37231 7/20 0.36
AKR1C3 P42330 2/20 0.35
AKR1C2 P52895 2/20 0.35
PTGS2 P35354 5/20 0.35
PTGS1 P23219 1/20 0.35
PPARA Q07869 3/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5558485 1.00 PPARG (0.36) PPARGAKR1C3AKR1C2PTGS2PTGS1
SCHEMBL5554636 0.91 POLB (0.36) PPARGAKR1C3AKR1C2PTGS2PPARA
SCHEMBL5559997 0.90 PPARG (0.33) PPARGAKR1C3AKR1C2PTGS2PPARA
SCHEMBL5558223 0.89 PTGS2 (0.35) AKR1C3AKR1C2PTGS2PTGS1
SCHEMBL5560462 0.84 PTGS2 (0.34) PPARGAKR1C3AKR1C2PTGS2PPARA
SCHEMBL5558544 0.84 PTGS2 (0.34) PPARGAKR1C3AKR1C2PTGS2PPARA
SCHEMBL5554459 0.81 PPARG (0.38) PPARGAKR1C3AKR1C2PTGS2PTGS1
SCHEMBL5554806 0.80 CNR2 (0.36) AKR1C3AKR1C2PTGS2POLB
SCHEMBL5558629 0.80 AKR1C3 (0.37) AKR1C3AKR1C2PTGS2POLB
SCHEMBL5800575 0.79 PTGS2 (0.43) PPARGAKR1C3AKR1C2PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
WO-2006050120-A2 SYNTHESIS OF COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2006-05-11 WO disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed