SCHEMBL5558830

SCHEMBL5558830

CC(=O)Oc1c(C)n(C(=O)c2ccc(C(F)(F)F)cc2)c2cc(Cl)c(O)c(C3CCCC3)c12

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 2/20 0.36
AKR1C2 P52895 1/20 0.36
SRC P12931 2/20 0.35
PRKACA P17612 2/20 0.35
PRKACG P22612 2/20 0.35
PRKACB P22694 2/20 0.35
MGLL Q99685 1/20 0.34
CNR1 P21554 1/20 0.34
CETP P11597 3/20 0.33
MAPK7 Q13164 1/20 0.33
MEN1 O00255 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
KMT2A Q03164 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
PROKR1 Q8TCW9 2/20 0.33
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
CCR1 P32246 1/20 0.32
CCR2 P41597 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5553945 0.90 PTGS2 (0.40) AKR1C3AKR1C2MEN1KMT2APTGDR2
SCHEMBL5558610 0.78 PTGS2 (0.43) AKR1C3AKR1C2MEN1KMT2APTGDR2
SCHEMBL5558391 0.77 SRC (0.42) AKR1C3AKR1C2SRCPRKACAPRKACG
SCHEMBL5558909 0.75 MAPK7 (0.39) MGLLMAPK7PTGS2
SCHEMBL5559277 0.75 SCN9A (0.37) MGLLMAPK7PTGS2
SCHEMBL5553718 0.75 PTGS2 (0.38) AKR1C3AKR1C2MEN1KMT2APTGDR2
SCHEMBL5560487 0.74 PDE2A (0.37) AKR1C3AKR1C2MGLLPTGS2
SCHEMBL5559446 0.74 MAPK7 (0.39) MGLLMAPK7PTGDR2
SCHEMBL5556641 0.71 ABCB11 (0.33) MAPK7HPGDKMT2APROKR1
SCHEMBL5559111 0.71 PPARG (0.40) AKR1C3AKR1C2MEN1KMT2APTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed