SCHEMBL5560487

SCHEMBL5560487

CC(=O)Oc1c(C)n(C(=O)c2ccc(Cl)c(F)c2)c2ccc(O)c(C3CCC3)c12

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 1/20 0.37
F10 P00742 1/20 0.32
TACR3 P29371 4/20 0.31
TACR2 P21452 3/20 0.31
TACR1 P25103 2/20 0.31
MAOB P27338 1/20 0.31
MGLL Q99685 3/20 0.31
PTGS2 P35354 2/20 0.31
KCNH2 Q12809 1/20 0.31
AKR1C3 P42330 1/20 0.30
AKR1C2 P52895 1/20 0.30
PARP1 P09874 1/20 0.30
PARP2 Q9UGN5 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5553718 0.87 PTGS2 (0.38) PTGS2AKR1C3AKR1C2
SCHEMBL5558954 0.85 CNR1 (0.37) MGLL
SCHEMBL5800435 0.85 MAOB (0.35) TACR3TACR2TACR1MAOBPTGS2
SCHEMBL5559110 0.81 MAOB (0.35) TACR3TACR2TACR1MAOBPTGS2
SCHEMBL5559277 0.79 SCN9A (0.37) MGLLPTGS2
SCHEMBL5560527 0.79 PTGS2 (0.33) MAOBPTGS2KCNH2AKR1C3AKR1C2
SCHEMBL5800516 0.78 ABCB11 (0.35) PTGS2AKR1C3AKR1C2
SCHEMBL5554202 0.78 TACR3 (0.33) TACR3TACR2TACR1MAOBPTGS2
SCHEMBL5559667 0.76 PTGS2 (0.35) PDE2ATACR3TACR2TACR1MAOB
SCHEMBL5800412 0.76 PTGS2 (0.46) MAOBPTGS2AKR1C3AKR1C2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1643961-A4 COX-2 AND FAAH INHIBITORS MICROBIA INC (US) 2007-09-12 EP disclosed
EP-1643961-A2 COX-2 AND FAAH INHIBITORS Microbia, Inc. (US) 2006-04-12 EP disclosed
WO-2005002525-A2 COX-2 AND FAAH INHIBITORS MICROBIA, INC. (US) 2005-01-13 WO disclosed