SCHEMBL5565742

SCHEMBL5565742

CCN(C(=O)c1ccc(C(=O)OC)s1)c1cccc(-c2cccs2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
ALDH1A1 P00352 1/20 0.46
HSD17B2 P37059 9/20 0.41
HSD17B1 P14061 8/20 0.41
MAPT P10636 2/20 0.40
NR4A2 P43354 1/20 0.40
NPSR1 Q6W5P4 3/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
ATM Q13315 1/20 0.38
PSMB5 P28074 1/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
PRMT6 Q96LA8 1/20 0.38
RXFP1 Q9HBX9 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5565995 0.90 KDM4E (0.48) KDM4ENPC1RAB9AALDH1A1HSD17B2
SCHEMBL5565065 0.80 NPSR1 (0.42) KDM4ERAB9AMAPTNPSR1L3MBTL1
SCHEMBL6455153 0.79 ALDH1A1 (0.50) KDM4EALDH1A1MAPTNPSR1L3MBTL1
SCHEMBL5563984 0.78 HSD17B2 (0.42) HSD17B2HSD17B1NPSR1L3MBTL1HPGD
SCHEMBL6462245 0.78 KDM4E (0.45) KDM4ENPC1RAB9AALDH1A1MAPT
SCHEMBL6454902 0.73 ALDH1A1 (0.46) KDM4EALDH1A1HSD17B2HSD17B1MAPT
SCHEMBL5565747 0.72 SMN1; SMN2 (0.50) NPC1RAB9AMAPTHDAC3HDAC1
SCHEMBL5564443 0.72 NPSR1 (0.46) ALDH1A1MAPTNPSR1L3MBTL1HPGD
SCHEMBL5557107 0.72 NPSR1 (0.43) ALDH1A1MAPTNPSR1L3MBTL1HPGD
SCHEMBL4579984 0.71 NPC1 (0.46) KDM4ENPC1RAB9AALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1778683-A1 THIOPHENE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-05-02 EP disclosed
WO-2005121134-A1 THIOPHENE DERIVATIVES, THEIR MANUFACTURE AND USE AS PHARMACEUTICAL AGENTS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO disclosed