SCHEMBL5567757

SCHEMBL5567757

CC(O)(c1ccc(NS(=O)(=O)c2cccc(Cl)c2Cl)cc1)C(F)(F)F

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 13/20 0.59
PGR P06401 1/20 0.54
RORA P35398 4/20 0.54
RORC P51449 3/20 0.54
NR1H2 P55055 2/20 0.54
NR1H4 Q96RI1 1/20 0.54
NR1H3 Q13133 1/20 0.48
RORB Q92753 1/20 0.47
ALDH1A1 P00352 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5569339 0.90 HSD11B1 (0.65) HSD11B1PGRRORARORCNR1H2
SCHEMBL13615019 0.84 PGR (0.62) HSD11B1PGRRORAALDH1A1
SCHEMBL13239427 0.80 HSD11B1 (0.80) HSD11B1
SCHEMBL31078033 0.80 RORA (0.68) HSD11B1PGRRORARORCNR1H2
SCHEMBL4597584 0.80 HSD11B1 (0.59) HSD11B1RORARORCNR1H2ALDH1A1
SCHEMBL13875335 0.78 PGR (0.65) PGRALDH1A1
SCHEMBL16497560 0.77 RORA (0.49) HSD11B1RORARORCNR1H2NR1H4
SCHEMBL14613673 0.76 IDH1 (0.61) HSD11B1
SCHEMBL10455160 0.76 PGR (0.75) PGRALDH1A1
SCHEMBL17483805 0.75 PGR (0.62) PGRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8076376-B2 Aniline sulfonamide derivatives and their uses AMGEN INC. 2011-12-13 US disclosed
US-8076376-B2 Aniline sulfonamide derivatives and their uses AMGEN INC. 2011-12-13 US disclosed
US-8076376-B2 Aniline sulfonamide derivatives and their uses AMGEN INC. 2011-12-13 US disclosed
WO-2007013929-A1 ANILINE SULFONAMIDE DERIVATIVES AND THEIR USES AMGEN INC. (US) 2007-02-01 WO disclosed
US-20070021502-A1 Aniline sulfonamide derivatives and their uses AMGEN INC. 2007-01-25 US disclosed
US-20070021502-A1 Aniline sulfonamide derivatives and their uses AMGEN INC. 2007-01-25 US disclosed
US-20070021502-A1 Aniline sulfonamide derivatives and their uses AMGEN INC. 2007-01-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070021502-A1 Aniline sulfonamide derivatives and their uses ARSA, SULT2A1, SULT1A1 HSD11B1 680/4885PGR 2186/4885RORA 904/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.