SCHEMBL5569357

SCHEMBL5569357

CN1CCCCN1c1ccc(NC(=O)C2(N)CC3CCC2C3)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.36
MAPT P10636 7/20 0.35
ALDH1A1 P00352 4/20 0.35
KDM4E B2RXH2 3/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
GAA P10253 2/20 0.35
GFER P55789 2/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C19 P33261 1/20 0.34
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
EPHX2 P34913 4/20 0.33
HTT P42858 1/20 0.33
CNR2 P34972 1/20 0.32
IDO1 P14902 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5565253 0.85 NPC1 (0.34) MAPTALDH1A1MEN1KMT2AGAA
SCHEMBL25383720 0.77 L3MBTL1 (0.47) TSHRMAPTMEN1KMT2AGAA
SCHEMBL5504268 0.67 F10 (0.48)
SCHEMBL26747648 0.62 SLC1A2 (0.37) TSHRSMN1; SMN2LMNA
SCHEMBL1632303 0.61 ALDH1A1 (0.33) TSHRALDH1A1HTTL3MBTL1
Hydrochloric Acid SCHEMBL1632301 0.60 ALDH1A1 (0.32) TSHRALDH1A1NPSR1SMN1; SMN2L3MBTL1
SCHEMBL2009762 0.60 THRB (0.35) TSHRALDH1A1SMN1; SMN2LMNA
SCHEMBL3733593 0.60 SLC6A4 (0.41)
SCHEMBL202772 0.60 SLC6A4 (0.41)
SCHEMBL9457723 0.60 THRB (0.35) TSHRALDH1A1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1748997-A1 SUBSTITUTED THIOPHENE-2-CARBOXYLIC ACID AMIDES, THE PRODUCTION THEREOF AND THE USE THEREOF AS DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2007-02-07 EP disclosed
WO-2005111013-A1 SUBSTITUTED THIOPHENE-2-CARBOXYLIC ACID AMIDES, THE PRODUCTION THEREOF AND THE USE THEREOF AS DRUGS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2005-11-24 WO disclosed