SCHEMBL5574807

SCHEMBL5574807

CC(C)Oc1ccc(-c2c(-c3ccc(C(F)(F)F)cn3)ccc3[nH]c(CO)c(Cl)c23)cc1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP3A5 P20815 1/20 0.34
SCN9A Q15858 4/20 0.33
PTGES O14684 2/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33
PTPN5 P54829 1/20 0.33
PPARD Q03181 1/20 0.33
MAP4K4 O95819 1/20 0.32
MCHR1 Q99705 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
BTK Q06187 1/20 0.32
KDM4E B2RXH2 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
PRKAB2 O43741 1/20 0.31
PRKAG1 P54619 1/20 0.31
PRKAA2 P54646 1/20 0.31
PRKAA1 Q13131 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5267329 0.85 MCHR1 (0.35) CYP1A2CYP3A4CYP3A5SCN9APTGES
SCHEMBL5272120 0.84 MCHR1 (0.34) CYP1A2CYP3A4CYP3A5SCN9APTGES
SCHEMBL5573963 0.84 CYP1A2 (0.34) CYP1A2CYP3A4CYP3A5SCN9APTGES
SCHEMBL5350625 0.84 CYP1A2 (0.34) CYP1A2CYP3A4CYP3A5SCN9APTGES
SCHEMBL5571402 0.83 KDM4E (0.43) CYP1A2PTGESPPARDMCHR1MEN1
SCHEMBL5338178 0.80 PTGES (0.33) SCN9APTGESPTPN5PPARDMCHR1
SCHEMBL5571416 0.80 MLYCD (0.38) PTGESPPARDMCHR1MEN1KMT2A
SCHEMBL5570207 0.79 GPR35 (0.36) CYP1A2CYP3A4CYP3A5ALOX5APFEN1
SCHEMBL5573431 0.79 MCHR1 (0.37) CYP1A2CYP3A4CYP3A5SCN9AALOX5AP
SCHEMBL5574783 0.78 KDM4E (0.44) CYP1A2PPARDMCHR1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1841736-A1 INDOLES USEFUL IN THE TREATMENT OF INFLAMMATION Biolipox AB (SE) 2007-10-10 EP disclosed
WO-2006077367-A1 INDOLES USEFUL IN THE TREATMENT OF INFLAMATION BIOLIPOX AB (SE) 2006-07-27 WO disclosed