SCHEMBL5585315

SCHEMBL5585315

Fc1ccc(COc2ccnc(N3CCNCC3)n2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.49
ALDH1A1 P00352 8/20 0.47
CYP3A4 P08684 8/20 0.47
CYP2C9 P11712 8/20 0.47
CYP1A2 P05177 7/20 0.47
HSD17B10 Q99714 6/20 0.47
CASP1 P29466 6/20 0.47
CASP7 P55210 6/20 0.47
PRMT5 O14744 1/20 0.46
ACHE P22303 1/20 0.45
HTR6 P50406 2/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA9 Q16790 1/20 0.45
USP2 O75604 6/20 0.44
CYP2C19 P33261 6/20 0.44
HIF1A Q16665 6/20 0.44
HPGD P15428 4/20 0.44
MAPK1 P28482 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL905849 0.87 ACHE (0.60) ADRB1ALDH1A1CYP3A4CYP2C9CYP1A2
Hydrochloric Acid SCHEMBL27512588 0.86 ACHE (0.58) ADRB1ALDH1A1CYP3A4CYP2C9CYP1A2
SCHEMBL5258581 0.78 ADRB1 (0.52) ADRB1ALDH1A1ACHEHPGDKDM4E
SCHEMBL3267135 0.76 HTR2C (0.65) ADRB1ALDH1A1CYP3A4CYP2C9CYP1A2
SCHEMBL30423191 0.76 ADRB1 (0.50) ADRB1ALDH1A1CYP1A2HSD17B10CASP1
SCHEMBL905866 0.76 HTR6 (0.51) ADRB1ACHEHTR6CA12CA1
SCHEMBL2792154 0.75 ADRB1 (0.55) ADRB1ALDH1A1CYP2C9CYP1A2HSD17B10
SCHEMBL20443370 0.75 ADRB1 (0.52) ADRB1ALDH1A1ACHEKDM4E
Hydrochloric Acid SCHEMBL5368905 0.74 ALDH1A1 (0.54) ADRB1ALDH1A1CYP2C9CYP1A2HSD17B10
Hydrochloric Acid SCHEMBL3275509 0.73 ADRB1 (0.54) ADRB1ALDH1A1CYP3A4CYP2C9CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7247633-B2 Pyrimidine compounds and their use BIOVITRUM AB (SE) 2007-07-24 US disclosed
US-20040014767-A1 Novel compounds and their use BIOVITRUM AB, A SWEDISH CORPORATION 2004-01-22 US disclosed
EP-1335907-A1 PIPERAZINYLPYRAZINE COMPOUNDS AS AGONIST OR ANTAGONIST OF SEROTONIN 5HT-2 RECEPTOR BIOVITRUM AB (SE) 2003-08-20 EP disclosed
US-6593330-B2 Central nervous system disorders; antiserotonine agents BIOVITRUM (SE) 2003-07-15 US disclosed
US-20020147200-A1 Novel compounds and their use PROXIMAGEN NEUROSCIENCE PLC (GB) 2002-10-10 US disclosed
WO-2002040456-A1 PIPERAZINYLPYRAZINE COMPOUNDS AS AGONIST OR ANTAGONIST OF SEROTONIN 5HT-2 RECEPTOR BIOVITRUM AB (SE) 2002-05-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020147200-A1 Novel compounds and their use BRIX1, UGT1A1, NR5A1 ADRB1 275/4885ALDH1A1 288/4885CYP3A4 295/4885
US-20040014767-A1 Novel compounds and their use BRIX1, UGT1A1, NR5A1 ADRB1 275/4885ALDH1A1 288/4885CYP3A4 295/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.