SCHEMBL5592894

SCHEMBL5592894

CCN(CC)C1CCN(Cc2ccc(C(=O)N(NCC(C)C)c3nc(C#N)ncc3Cl)cc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.45
CTSB P07858 1/20 0.45
CTSS P25774 1/20 0.45
CTSK P43235 1/20 0.45
ACVR1 Q04771 1/20 0.39
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
CHRM2 P08172 2/20 0.36
PRKAA2 P54646 2/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CHRM4 P08173 1/20 0.35
OPRD1 P41143 3/20 0.35
OPRM1 P35372 2/20 0.34
OPRK1 P41145 2/20 0.34
CHRM3 P20309 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592691 0.88 CTSS (0.49) CTSLCTSBCTSSCTSK
SCHEMBL5593156 0.84 CTSL (0.43) CTSLCTSBCTSSCTSKFNTA
SCHEMBL5592803 0.83 CTSS (0.41) CTSLCTSBCTSSCTSKPRKAA2
SCHEMBL5592735 0.83 CTSS (0.49) CTSLCTSBCTSSCTSK
SCHEMBL8236817 0.83 CTSL (0.65) CTSLCTSBCTSSCTSKACVR1
SCHEMBL5592660 0.83 CTSS (0.49) CTSLCTSBCTSSCTSKCHRM2
Trifluoroacetic Acid SCHEMBL5592759 0.83 CTSL (0.47) CTSLCTSBCTSSCTSK
Trifluoroacetic Acid SCHEMBL5592942 0.82 CTSS (0.47) CTSLCTSBCTSSCTSKCHRM4
Trifluoroacetic Acid SCHEMBL5592645 0.81 CTSS (0.47) CTSLCTSBCTSSCTSKACVR1
Trifluoroacetic Acid SCHEMBL5592864 0.81 CTSS (0.47) CTSLCTSBCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025775-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed