SCHEMBL5593156

SCHEMBL5593156

CC(C)CNN(C(=O)c1ccc(CN2CCC(OC(=O)C(F)(F)F)CC2)cc1)c1nc(C#N)ncc1Cl

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
PRKAA2 P54646 11/20 0.35
PRKAB2 O43741 6/20 0.34
PRKAG1 P54619 6/20 0.34
PRKAA1 Q13131 6/20 0.34
PRKAG3 Q9UGI9 6/20 0.34
PRKAG2 Q9UGJ0 6/20 0.34
PRKAB1 Q9Y478 6/20 0.34
CYP3A4 P08684 1/20 0.34
CXCR3 P49682 1/20 0.34
MCHR1 Q99705 1/20 0.34
FNTA P49354 1/20 0.34
FNTB P49356 1/20 0.34
BCHE P06276 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5592942 0.85 CTSS (0.47) CTSLCTSBCTSSCTSKCXCR3
SCHEMBL5592691 0.85 CTSS (0.49) CTSLCTSBCTSSCTSKMCHR1
SCHEMBL5592894 0.84 CTSL (0.45) CTSLCTSBCTSSCTSKPRKAA2
Trifluoroacetic Acid SCHEMBL5592645 0.84 CTSS (0.47) CTSLCTSBCTSSCTSKMCHR1
Trifluoroacetic Acid SCHEMBL5592759 0.84 CTSL (0.47) CTSLCTSBCTSSCTSK
Trifluoroacetic Acid SCHEMBL5592864 0.83 CTSS (0.47) CTSLCTSBCTSSCTSKCYP3A4
SCHEMBL3168730 0.80 CTSL (0.44) CTSLCTSBCTSSCTSKPRKAA2
SCHEMBL5592803 0.80 CTSS (0.41) CTSLCTSBCTSSCTSKPRKAA2
SCHEMBL5592735 0.80 CTSS (0.49) CTSLCTSBCTSSCTSKMCHR1
SCHEMBL5592660 0.80 CTSS (0.49) CTSLCTSBCTSSCTSKPRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025775-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed